SCHEMBL8200346

SCHEMBL8200346

CCCCCCC1CCc2cc(C(=O)NCC3CCCC3(C)C)ccc2C1=O

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SGPL1 O95470 1/20 0.41
S1PR1 P21453 1/20 0.41
THRA P10827 1/20 0.39
THRB P10828 1/20 0.39
SMYD3 Q9H7B4 2/20 0.36
ITGB3 P05106 2/20 0.35
ITGA2B P08514 2/20 0.35
MAPK14 Q16539 3/20 0.34
HTR4 Q13639 1/20 0.33
CYP26A1 O43174 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199670 0.80 HTR2C (0.43)
SCHEMBL8192821 0.79 THRA (0.42) SGPL1S1PR1THRATHRBSMYD3
SCHEMBL8200249 0.77 THRA (0.52) SGPL1S1PR1THRATHRBITGB3
SCHEMBL8205603 0.77 SMN1; SMN2 (0.48) MAPK14
SCHEMBL8192695 0.77 THRA (0.49) SGPL1S1PR1THRATHRBITGB3
SCHEMBL8199839 0.75 MLYCD (0.45) SGPL1S1PR1THRATHRB
SCHEMBL18052663 0.70 THRA (0.53) SGPL1S1PR1THRATHRBCYP26A1
SCHEMBL8201692 0.70 MLYCD (0.42) SGPL1S1PR1THRBITGB3ITGA2B
SCHEMBL15954361 0.69 THRA (0.52) SGPL1S1PR1THRATHRBCYP26A1
SCHEMBL15954358 0.69 THRA (0.52) SGPL1S1PR1THRATHRBCYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed