SCHEMBL8199839

SCHEMBL8199839

CCCCCCC1CCc2cc(C(=O)NCc3cc(C(F)(F)F)cc(C(F)(F)F)c3)ccc2C1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.45
HPGD P15428 6/20 0.44
ALDH1A1 P00352 6/20 0.44
KDM4E B2RXH2 4/20 0.44
GAA P10253 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
ROCK2 O75116 3/20 0.39
NAMPT P43490 1/20 0.39
THRA P10827 1/20 0.39
THRB P10828 1/20 0.39
P2RX1 P51575 1/20 0.38
TMPRSS4 Q9NRS4 1/20 0.38
SGPL1 O95470 1/20 0.38
S1PR1 P21453 1/20 0.38
CCR2 P41597 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200677 0.83 MLYCD (0.47) MLYCDHPGDALDH1A1KDM4EGAA
SCHEMBL8192821 0.81 THRA (0.42) MLYCDALDH1A1NAMPTTHRATHRB
SCHEMBL8205603 0.79 SMN1; SMN2 (0.48) ALDH1A1CYP1A2CYP2D6CYP2C19CYP2C9
SCHEMBL8200249 0.77 THRA (0.52) THRATHRBSGPL1S1PR1
SCHEMBL8192695 0.77 THRA (0.49) ALDH1A1NPSR1THRATHRBSGPL1
SCHEMBL8200346 0.75 SGPL1 (0.41) THRATHRBSGPL1S1PR1
SCHEMBL8200629 0.74 P2RX1 (0.45) MLYCDHPGDKDM4EP2RX1TMPRSS4
SCHEMBL8201692 0.72 MLYCD (0.42) MLYCDNAMPTTHRBSGPL1S1PR1
SCHEMBL18052663 0.70 THRA (0.53) THRATHRBSGPL1S1PR1
SCHEMBL15954358 0.69 THRA (0.52) THRATHRBSGPL1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed