SCHEMBL8200677

SCHEMBL8200677

C=CCC1CCc2cc(C(=O)NCc3cc(C(F)(F)F)cc(C(F)(F)F)c3)ccc2C1=O

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 2/20 0.47
ALDH1A1 P00352 6/20 0.42
KDM4E B2RXH2 4/20 0.42
CCR2 P41597 2/20 0.42
HPGD P15428 6/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
ROCK2 O75116 2/20 0.41
NAMPT P43490 1/20 0.41
P2RX1 P51575 1/20 0.40
TMPRSS4 Q9NRS4 1/20 0.40
GAA P10253 2/20 0.40
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199839 0.83 MLYCD (0.45) MLYCDALDH1A1KDM4ECCR2HPGD
SCHEMBL8205119 0.81 CCR2 (0.45) MLYCDCCR2HPGDP2RX1TMPRSS4
SCHEMBL8198845 0.79 MLYCD (0.40) MLYCDNAMPTITGB3ITGA2B
SCHEMBL8199811 0.76 CYP26A1 (0.47) ALDH1A1ITGB3ITGA2B
SCHEMBL14061976 0.70 CYP26A1 (0.64) ALDH1A1CYP1A2CYP2D6CYP2C19CYP3A4
SCHEMBL14173369 0.68 MLYCD (0.47) MLYCDALDH1A1KDM4ECCR2HPGD
SCHEMBL8199804 0.68 HTR2C (0.49) ALDH1A1CCR2GAA
SCHEMBL17211818 0.67 METAP1 (0.48)
SCHEMBL22517021 0.67 ITGB3 (0.55) ALDH1A1ITGB3ITGA2B
SCHEMBL14061945 0.67 CYP24A1 (0.49) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed