SCHEMBL8201582

SCHEMBL8201582

COc1ccc(S(=O)(=O)n2cc(C(C)C3CCCN3)c3cc(Cl)ccc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 17/20 0.50
KDM1A O60341 1/20 0.42
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 2/20 0.41
HTR2A P28223 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
DRD2 P14416 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2C P28335 1/20 0.41
SLC6A4 P31645 1/20 0.41
HTR7 P34969 1/20 0.41
HRH1 P35367 1/20 0.41
ADRA1B P35368 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208598 0.89 HTR6 (0.48) HTR6KDM1AKCNH2
SCHEMBL8209521 0.89 HTR6 (0.51) HTR6KDM1A
SCHEMBL8201576 0.87 HTR6 (0.63) HTR6
SCHEMBL8208098 0.87 HTR6 (0.48) HTR6CYP3A4CYP2D6HTR2A
SCHEMBL8201606 0.81 HTR6 (0.45) HTR6HTR2ADRD2HTR7
SCHEMBL8201598 0.80 AKR1C3 (0.46)
SCHEMBL8208544 0.80 HTR6 (0.44) HTR6KDM1A
SCHEMBL8201465 0.79 HTR6 (0.43) HTR6HTR2ADRD2
SCHEMBL8209795 0.79 HTR6 (0.49) HTR6KDM1ACYP3A4CYP2D6
SCHEMBL7472995 0.79 HTR6 (0.48) HTR6KDM1ACYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100291-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-08 US claimed
WO-1999047516-A1 3-(2-PYRROLIDINYLMETHYL)-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY SLASSI ABDELMALIK (CA) 1999-09-23 WO claimed
US-6100291-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-08 US disclosed
WO-1999047516-A1 3-(2-PYRROLIDINYLMETHYL)-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY SLASSI ABDELMALIK (CA) 1999-09-23 WO disclosed