SCHEMBL8202408

SCHEMBL8202408

O=C1NC2=C(CCC=C2)Oc2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.36
GSK3B P49841 1/20 0.36
PLA2G1B P04054 1/20 0.34
ATG4B Q9Y4P1 1/20 0.34
LMNA P02545 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
MAPT P10636 4/20 0.33
CASP3 P42574 2/20 0.33
CASP7 P55210 2/20 0.33
CASP6 P55212 2/20 0.33
CASP8 Q14790 2/20 0.33
TDP2 O95551 1/20 0.33
CASP9 P55211 1/20 0.33
MAP3K14 Q99558 1/20 0.33
CASP2 P42575 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18222130 0.80 ALOX5 (0.48) KDM4ELMNATDP1MAPTL3MBTL1
SCHEMBL8796463 0.69 CASP7 (0.44) KDM4EALDH1A1GSK3BLMNAMAPT
SCHEMBL4490831 0.69 LRRK2 (0.51) KDM4EALDH1A1GSK3BLMNAMAPT
SCHEMBL380110 0.65 ALOX5 (0.61) KDM4EALDH1A1GSK3BLMNATDP1
SCHEMBL16306320 0.63 KDM4E (0.53) KDM4EALDH1A1GSK3BLMNATDP1
SCHEMBL17452157 0.63 CA1 (0.33) ALDH1A1KMT2A
SCHEMBL11168286 0.62 ACVR1 (0.41) GSK3BMAPTL3MBTL1PDGFRAFER
SCHEMBL23175285 0.60 CA12 (0.52) KDM4EALDH1A1GSK3BLMNATDP1
SCHEMBL6171749 0.60 CASP3 (0.53) KDM4EALDH1A1GSK3BLMNATDP1
SCHEMBL19888558 0.60 KDM4E (0.34) KDM4EPKMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2489657-A2 Inhibitors of histone deacetylase MethylGene Inc. (CA) 2012-08-22 EP disclosed
WO-2009137499-A1 INHIBITORS OF HISTONE DEACETYLASE ENVIVO PHARMACEUTICALS, INC. (US) 2009-11-12 WO disclosed
WO-2008055068-A2 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2008-05-08 WO disclosed