SCHEMBL8202767

SCHEMBL8202767

O=C(NCc1cccc2ccccc12)c1ccc2c(c1)CCC(CCN1CCC(c3ccccc3)CC1)C2=O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.44
DRD2 P14416 4/20 0.42
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
P2RX7 Q99572 1/20 0.40
MCHR1 Q99705 1/20 0.39
TGM2 P21980 1/20 0.38
CA2 P00918 1/20 0.38
PPARG P37231 1/20 0.38
HTR1A P08908 3/20 0.38
HTR2A P28223 3/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8202309 0.92 HTR2C (0.43) HTR2CDRD2HTR1DHTR1BOPRM1
SCHEMBL8199804 0.89 HTR2C (0.49) HTR2CDRD2OPRM1OPRK1MCHR1
SCHEMBL8202320 0.85 USP5 (0.52) HTR2CDRD2MCHR1
SCHEMBL8588802 0.83 HTR2C (0.48) HTR2CDRD2OPRM1OPRK1MCHR1
SCHEMBL8202304 0.83 HTR2C (0.47) HTR2CDRD2MCHR1
SCHEMBL8198570 0.83 HTR2C (0.47) HTR2CDRD2OPRM1OPRK1HTR2A
SCHEMBL8199074 0.82 HTR2C (0.48) HTR2CDRD2OPRM1OPRK1MCHR1
SCHEMBL8204772 0.82 HTR2C (0.50) HTR2CDRD2MCHR1
SCHEMBL8200236 0.82 DRD2 (0.40) HTR2CDRD2OPRM1OPRK1MCHR1
SCHEMBL8199695 0.82 SLC6A2 (0.46) HTR2CDRD2OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed