SCHEMBL8200236

SCHEMBL8200236

O=C(NCCc1cccc2c1oc1ccccc12)c1ccc2c(c1)CCC(CCN1CCC(c3ccccc3)CC1)C2=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.40
HTR2A P28223 10/20 0.40
HTR1A P08908 4/20 0.40
HTR2C P28335 3/20 0.40
DRD3 P35462 6/20 0.40
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
MAOB P27338 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRK1 P41145 1/20 0.35
MCHR1 Q99705 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8202309 0.88 HTR2C (0.43) DRD2HTR2AHTR1AHTR2CDRD3
SCHEMBL8199074 0.85 HTR2C (0.48) DRD2HTR2COPRM1OPRK1MCHR1
SCHEMBL8198570 0.84 HTR2C (0.47) DRD2HTR2AHTR2COPRM1OPRK1
SCHEMBL8199919 0.83 ADRA2A (0.48) BCHEACHE
SCHEMBL8588802 0.83 HTR2C (0.48) DRD2HTR2CDRD3OPRM1OPRK1
SCHEMBL8202767 0.82 HTR2C (0.44) DRD2HTR2AHTR1AHTR2COPRM1
SCHEMBL8191625 0.82 DRD2 (0.44) DRD2HTR2CDRD3
SCHEMBL8198781 0.81 HTR2C (0.46) DRD2HTR2CDRD3MCHR1
SCHEMBL8200603 0.81 HTR2C (0.49) DRD2HTR2AHTR2C
SCHEMBL8199804 0.81 HTR2C (0.49) DRD2HTR2COPRM1OPRK1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed