SCHEMBL8203738

SCHEMBL8203738

CSCC[C@H](NC(=O)OC(C)(C)C)C(C)=O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.64
CTSS P25774 4/20 0.64
CA2 P00918 1/20 0.49
TSHR P16473 1/20 0.48
EPHX2 P34913 1/20 0.47
ALDH1A1 P00352 4/20 0.46
LMNA P02545 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 4/20 0.44
MAPT P10636 1/20 0.44
KLK7 P49862 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
HPGD P15428 2/20 0.42
THRB P10828 1/20 0.42
KLK5 Q9Y337 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13778725 1.00 CTSK (0.64) CTSKCTSSCA2TSHREPHX2
SCHEMBL15081482 1.00 CTSK (0.64) CTSKCTSSCA2TSHREPHX2
SCHEMBL6623782 0.89 CTSK (0.63) CTSKCTSSCA2TSHREPHX2
SCHEMBL6623780 0.89 CTSK (0.63) CTSKCTSSCA2TSHREPHX2
SCHEMBL5717952 0.89 CTSK (0.63) CTSKCTSSCA2TSHREPHX2
SCHEMBL17326876 0.88 CTSS (0.56) CTSKCTSSCA2
SCHEMBL352156 0.87 CTSS (0.68) CTSKCTSSCA2TSHREPHX2
SCHEMBL478905 0.87 CTSS (0.68) CTSKCTSSCA2TSHREPHX2
SCHEMBL4395744 0.87 CTSS (0.68) CTSKCTSSCA2TSHREPHX2
SCHEMBL27704332 0.87 CTSK (0.64) CTSKCTSSCA2TSHREPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015140481-A1 ANTIMICROBIAL COMPOUNDS bioMérieux (FR) 2015-09-24 WO disclosed
EP-1054865-A1 FARNESYL TRANSFERASE INHIBITORS AstraZeneca UK Limited (GB) 2000-11-29 EP disclosed
WO-1999041235-A1 FARNESYL TRANSFERASE INHIBITORS ASTRAZENECA UK LIMITED (GB) 1999-08-19 WO disclosed