SCHEMBL478905

SCHEMBL478905

CSCCC(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.68
CTSK P43235 4/20 0.68
TSHR P16473 2/20 0.54
CA2 P00918 1/20 0.49
LMNA P02545 1/20 0.48
PPARG P37231 3/20 0.47
PPARA Q07869 3/20 0.47
KLK7 P49862 1/20 0.47
EPHX2 P34913 1/20 0.47
USP2 O75604 1/20 0.46
MAPK1 P28482 1/20 0.46
PPARD Q03181 2/20 0.45
ALDH1A1 P00352 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
KLK5 Q9Y337 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL352156 1.00 CTSS (0.68) CTSSCTSKTSHRCA2LMNA
SCHEMBL4395744 1.00 CTSS (0.68) CTSSCTSKTSHRCA2LMNA
SCHEMBL1486229 1.00 CTSS (0.68) CTSSCTSKTSHRCA2LMNA
Methanesulfonamide SCHEMBL6898028 0.92 CTSS (0.60) CTSSCTSKTSHRCA2LMNA
Methanesulfonamide SCHEMBL6777577 0.92 CTSS (0.60) CTSSCTSKTSHRCA2LMNA
SCHEMBL2118282 0.90 CTSK (0.56) CTSSCTSKTSHRCA2PPARG
SCHEMBL2118283 0.90 CTSK (0.56) CTSSCTSKTSHRCA2PPARG
SCHEMBL7874195 0.89 CTSS (0.57) CTSSCTSKTSHRCA2LMNA
SCHEMBL7874192 0.89 CTSS (0.57) CTSSCTSKTSHRCA2LMNA
SCHEMBL16715127 0.89 CTSK (0.56) CTSSCTSKTSHRCA2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 408 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10000520-B2 B-vitamin and amino acid conjugates ofnicotinoyl ribosides and reduced nicotinoyl ribosides, derivatives thereof, and methods of preparation thereof ChromaDex Inc. (US) 2018-06-19 US claimed
CN-107708432-A Rumen bypass animal feed composition and preparation method thereof 拜内梅尔克公司 2018-02-16 CN claimed
US-20170267709-A1 B-VITAMIN AND AMINO ACID CONJUGATES OFNICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, DERIVATIVES THEREOF, AND METHODS OF PREPARATION THEREOF ChromaDex Inc. (US) 2017-09-21 US claimed
CN-103421087-A Liquid-phase synthesizing method for polypeptide SHANGHAI BAJIAYI PHARMACEUTICAL TECHNOLOGY CO LTD 2013-12-04 CN claimed
CN-102775591-A Preparation method of tetraamino-terminated glycolide-lactide telechelic copolymer UNIV HEBEI SCIENCE & TECH 2012-11-14 CN claimed
CN-1241935-C Liquid phase sgnthesis method of thymus pentapeptide UNIV LANZHOU (CN) 2006-02-15 CN claimed
CN-1634975-A Process for preparing 2,4-synthetic antigen with added spacing arms UNIV TSINGHUA (CN) 2005-07-06 CN claimed
CN-1513872-A Liquid phase sgnthesis method of thymus pentapeptide 兰州大学 2004-07-21 CN claimed
US-12625431-B2 EUV resist underlayer film-forming composition NISSAN CHEMICAL CORPORATION (JP) 2026-05-12 US disclosed
US-12617782-B2 Pyridazinones as PARP7 inhibitors RIBON THERAPEUTICS, INC. (US) 2026-05-05 US disclosed
EP-4142732-B1 METHODS OF USE FOR PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS INC (US) 2026-04-22 EP disclosed
US-12516063-B2 Substituted 7-(methylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide derivatives for treating autoimmune diseases ELI LILLY AND COMPANY (US) 2026-01-06 US disclosed
EP-3966226-B1 MASP INHIBITORY COMPOUNDS AND USES THEREOF BAYER AG (DE) 2025-12-24 EP disclosed
US-12503491-B2 MASP inhibitory compounds and uses thereof BAYER AKTIENGESELLSCHAFT (DE) 2025-12-23 US disclosed
US-5430052-A Protective effect against myocardial disorders caused by calcium ion overload; antiischemic agents; remedy for heart failure, angina pectoris NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1995-07-04 US disclosed
CN-1066070-A Promote the new benzo-fused lactams that tethelin discharges MERCK & CO INC (US) 1992-11-11 CN disclosed
EP-0467856-A2 Aminoalkanesulfonic acid derivatives and pharmaceutical compositions for use in preventing or treating heart diseases NIPPON ZOKI PHARMACEUTICAL CO. LTD. (JP) 1992-01-22 EP disclosed
EP-0376040-A2 N-phosphinyl di-and tripeptides as renin inhibitors AMERICAN CYANAMID COMPANY (US) 1990-07-04 EP disclosed
EP-0186977-A2 Renin-inhibitory dipeptides, their preparation and use SANKYO COMPANY LIMITED (JP) 1986-07-09 EP disclosed
US-3968226-A 3-Heterocyclic thiomethylcephalosporins as antibacterial agents SMITHKLINE CORPORATION (US) 1976-07-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12503491-B2 MASP inhibitory compounds and uses thereof MASP2, SERPINB1, SPINT2 CTSS 138/4885CTSK 149/4885TSHR 3032/4885
US-10000520-B2 B-vitamin and amino acid conjugates ofnicotinoyl ribosides and reduced nicotinoyl ribosides, derivatives thereof, and methods of preparation thereof NAMPT, NAPRT, NNMT CTSS 4478/4885CTSK 4555/4885TSHR 833/4885
US-12625431-B2 EUV resist underlayer film-forming composition EEF1A1, ARF1, EMG1 CTSS 4528/4885CTSK 3728/4885TSHR 3840/4885
US-12617782-B2 Pyridazinones as PARP7 inhibitors PARP3, PARP2, PARP1 CTSS 1086/4885CTSK 1225/4885TSHR 371/4885
US-20170267709-A1 B-VITAMIN AND AMINO ACID CONJUGATES OFNICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, DERIVATIVES THEREOF, AND METHODS OF PREPARATION THEREOF NAMPT, NAPRT, NNMT CTSS 4478/4885CTSK 4555/4885TSHR 833/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.