SCHEMBL8204875

SCHEMBL8204875

CN(C)c1nccc2c1CN(C(=O)O)C2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.34
ALDH1A1 P00352 2/20 0.34
NOTUM Q6P988 1/20 0.32
SORD Q00796 1/20 0.31
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31
HSD17B10 Q99714 2/20 0.30
PROKR1 Q8TCW9 2/20 0.30
ADRB2 P07550 1/20 0.30
GRIN2D O15399 1/20 0.30
GRIN3B O60391 1/20 0.30
CHRM1 P11229 1/20 0.30
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2A Q12879 1/20 0.30
GRIN2B Q13224 1/20 0.30
GRIN2C Q14957 1/20 0.30
GRIN3A Q8TCU5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17624117 0.76 USP2 (0.36) ALDH1A1HSD17B10GRIN2DGRIN3BCHRM1
SCHEMBL2806211 0.74 P2RX7 (0.32) CYP1A2CYP3A4CLK4
SCHEMBL22582925 0.73 UCHL1 (0.33) KDM4EALDH1A1
SCHEMBL13223182 0.72 ATM (0.33)
SCHEMBL8194629 0.72 NOTUM (0.41) KDM4EALDH1A1NOTUMMEN1KMT2A
SCHEMBL7946982 0.67 TRAP1 (0.52) ALDH1A1NOTUMMEN1KMT2ACYP3A4
SCHEMBL3722963 0.67 LMNA (0.34) HSD17B10
SCHEMBL16269004 0.67 NOTUM (0.39) KDM4ENOTUMMEN1KMT2ANLRP3
SCHEMBL28886631 0.66 KDM4E (0.31) KDM4EALDH1A1
SCHEMBL8193162 0.65 NAMPT (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033389-A2 MACROCYCLIC HCV INHIBITORS AND THEIR USES NOVARTIS AG (CH) 2008-03-20 WO disclosed