SCHEMBL8210848

SCHEMBL8210848

O=c1cccc(O)cc1-c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.55
HDAC2 Q92769 2/20 0.55
HDAC8 Q9BY41 2/20 0.55
HDAC6 Q9UBN7 1/20 0.55
ALOX5 P09917 1/20 0.52
BACE1 P56817 1/20 0.48
HSD17B1 P14061 4/20 0.47
ESR2 Q92731 3/20 0.47
ESR1 P03372 2/20 0.47
HSD17B2 P37059 3/20 0.47
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 1/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
MPI P34949 1/20 0.46
KMT2A Q03164 1/20 0.46
CA12 O43570 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15437890 0.77 HDAC4 (0.62) HDAC4HDAC2HDAC8HDAC6BACE1
SCHEMBL5389905 0.77 HDAC4 (0.62) HDAC4HDAC2HDAC8HDAC6BACE1
SCHEMBL2442343 0.77 GSTP1 (0.62) HDAC4HDAC2HDAC8HDAC6ALOX5
SCHEMBL5050883 0.76 HSD17B1 (0.58) ALOX5BACE1HSD17B1ESR2ESR1
SCHEMBL8450704 0.75 ALOX5 (0.63) ALOX5BACE1HSD17B1ESR2ESR1
SCHEMBL7616374 0.74 HDAC4 (0.65) HDAC4HDAC2HDAC8HDAC6BACE1
Biphenyl SCHEMBL18315407 0.74 CYP3A4 (0.71) ALOX5BACE1HSD17B1ESR2ESR1
SCHEMBL4651426 0.74 HSD17B1 (0.56) ALOX5BACE1HSD17B1ESR2ESR1
SCHEMBL10481639 0.73 HDAC4 (0.77) HDAC4HDAC2HDAC8HDAC6BACE1
SCHEMBL11328974 0.73 ALDH1A1 (0.57) HDAC4HDAC2HDAC8HDAC6ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096144-A TREATING WITH ACIDIC OR ALKALINE SOLUTION OF CONJUGATED UNSATURATED COMPOUND WITH AT LEAST 5 BONDS SHIN-ETSU CHEMICAL CO., LTD. (JP) 2000-08-01 US disclosed
US-5858571-A TREATING A PULVERIZED HYDROGEN ABSORBING ALLOY WITH A SOLUTION COMPRISING A CONJUGATED UNSATURATED COMPOUND SHIN-ETSU CHEMICAL CO., LTD. (JP) 1999-01-12 US disclosed