SCHEMBL8215899

SCHEMBL8215899

O=C1C(Br)=C(c2ccccc2)c2ccc(O)cc21

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 16/20 0.69
ESR1 P03372 15/20 0.69
MAOA P21397 1/20 0.50
UGT1A1 P22309 1/20 0.50
MAOB P27338 1/20 0.50
ALOX5 P09917 1/20 0.47
P2RX7 Q99572 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8234582 0.84 ESR2 (0.62) ESR2ESR1MAOAUGT1A1MAOB
SCHEMBL8242608 0.84 ESR2 (0.62) ESR2ESR1MAOAUGT1A1MAOB
SCHEMBL8236050 0.83 ESR2 (0.50) ESR2ESR1MAOAUGT1A1MAOB
SCHEMBL3922937 0.81 ESR2 (1.00) ESR2ESR1MAOAUGT1A1MAOB
SCHEMBL8242350 0.81 ESR2 (0.54) ESR2ESR1MAOAUGT1A1MAOB
SCHEMBL8235168 0.80 ESR2 (0.57) ESR2ESR1MAOAUGT1A1MAOB
SCHEMBL5139553 0.80 FGFR1 (0.55) MAOAP2RX7
SCHEMBL8246534 0.80 ESR2 (0.49) ESR2ESR1MAOAUGT1A1MAOB
SCHEMBL3575957 0.79 FGFR1 (0.70) ESR2ESR1MAOAUGT1A1MAOB
SCHEMBL8927863 0.76 ESR2 (0.65) ESR2ESR1MAOAUGT1A1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8877747-B2 Indenone derivative and pharmaceutical composition comprising same KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2014-11-04 US disclosed
US-8877747-B2 Indenone derivative and pharmaceutical composition comprising same KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2014-11-04 US disclosed
US-8877747-B2 Indenone derivative and pharmaceutical composition comprising same KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2014-11-04 US disclosed
EP-2475649-B1 INDENONE DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME KOREA RES INST CHEM TECH (KR) 2014-08-13 EP disclosed
EP-2475649-B1 INDENONE DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME KOREA RES INST CHEM TECH (KR) 2014-08-13 EP disclosed
US-20120214991-A1 Indenone Derivative and Pharmaceutical Composition Comprising Same KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2012-08-23 US disclosed
US-20120214991-A1 Indenone Derivative and Pharmaceutical Composition Comprising Same KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2012-08-23 US disclosed
US-20120214991-A1 Indenone Derivative and Pharmaceutical Composition Comprising Same KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2012-08-23 US disclosed
EP-2475649-A1 INDENONE DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME Korea Research Institute Of Chemical Technology (KR) 2012-07-18 EP disclosed
WO-2011030955-A1 INDENONE DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2011-03-17 WO disclosed
WO-2011030955-A1 INDENONE DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2011-03-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120214991-A1 Indenone Derivative and Pharmaceutical Composition Comprising Same INSR, HSD17B7, SOST ESR2 325/4885ESR1 1113/4885MAOA 3574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.