SCHEMBL8219366

SCHEMBL8219366

[c]1ccc(N2CCC(=NN3CCOCC3)CC2)nc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.33
HPGD P15428 4/20 0.33
HSD17B10 Q99714 4/20 0.33
KDM4E B2RXH2 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
AKR1C3 P42330 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
RECQL P46063 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
LRRK2 Q5S007 1/20 0.32
CNR2 P34972 3/20 0.32
POLB P06746 1/20 0.30
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL182759 0.82 ALDH1A1 (0.44) ALDH1A1HPGDHSD17B10KDM4ESMN1; SMN2
SCHEMBL8197207 0.77 GAA (0.33) GAA
SCHEMBL8194012 0.76 ADK (0.43)
SCHEMBL8219361 0.75 LRRK2 (0.30) LRRK2
SCHEMBL8219363 0.75 LRRK2 (0.30) LRRK2
SCHEMBL4775116 0.71 LMNA (0.36) LMNA
SCHEMBL743397 0.70 MAPT (0.40) ALDH1A1SMN1; SMN2CYP1A2LMNAMAPT
SCHEMBL2067822 0.70 MAPT (0.36) ALDH1A1KDM4ESMN1; SMN2CYP1A2LMNA
SCHEMBL8192471 0.70 GPR119 (0.32)
SCHEMBL4778875 0.70 HRH3 (0.37) KDM4ECYP1A2MEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000023444-A1 5,7-DISUBSTITUTED-4-AMINOPYRIDO[2,3-D]PYRIMIDINE COMPOUNDS ABBOTT LABORATORIES (US) 2000-04-27 WO claimed
WO-2000023444-A1 5,7-DISUBSTITUTED-4-AMINOPYRIDO[2,3-D]PYRIMIDINE COMPOUNDS ABBOTT LABORATORIES (US) 2000-04-27 WO disclosed