SCHEMBL8225299

SCHEMBL8225299

F[C@@]1(CNC2CC2)CNC[C@H]1Cc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
GBA1 P04062 2/20 0.36
GRIN2B Q13224 2/20 0.34
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
BACE1 P56817 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3910560 1.00 MEN1 (0.37) MEN1RAB9AKMT2AGBA1GRIN2B
SCHEMBL8222794 0.79 GBA1 (0.40) GBA1SLC6A2SLC6A4SLC6A3
SCHEMBL8225218 0.69 GBA1 (0.37) GBA1SLC6A2SLC6A4SLC6A3
SCHEMBL27475180 0.66 GBA1 (0.51) GBA1
SCHEMBL8222704 0.65 GBA1 (0.51) MEN1RAB9AKMT2AGBA1GRIN2B
SCHEMBL3913849 0.65 GBA1 (0.51) MEN1RAB9AKMT2AGBA1GRIN2B
SCHEMBL8225319 0.63 OPRM1 (0.44) MEN1RAB9AKMT2ASLC6A2SLC6A4
SCHEMBL663239 0.61 GRIN2B (0.74) MEN1RAB9AKMT2AGRIN2BBCHE
SCHEMBL25698481 0.60 NOS3 (0.40) GBA1
SCHEMBL3910981 0.60 GBA1 (0.49) GBA1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007140980-A1 PYRROLIDINE DERIVATIVES USEFUL AS BACE INHIBITORS NOVARTIS AG (CH) 2007-12-13 WO disclosed