SCHEMBL8235167

SCHEMBL8235167

O=C1NCCN1c1cc[c]cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.40
CYP1A2 P05177 3/20 0.38
CYP3A4 P08684 3/20 0.38
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CRBN Q96SW2 1/20 0.36
MAP3K5 Q99683 1/20 0.35
SCN9A Q15858 1/20 0.35
CCNT1 O60563 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
CCND3 P30281 1/20 0.34
CDK7 P50613 1/20 0.34
CDK9 P50750 1/20 0.34
CCNH P51946 1/20 0.34
MNAT1 P51948 1/20 0.34
CDK6 Q00534 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30702779 0.74 CRBN (0.63) CYP3A4TSHRSMN1; SMN2HSD17B10CRBN
SCHEMBL2198674 0.74 CRBN (0.63) CYP3A4TSHRSMN1; SMN2HSD17B10CRBN
SCHEMBL3032630 0.73 MAP3K5 (0.38) TDO2CYP1A2CYP3A4TSHRSMN1; SMN2
SCHEMBL37681 0.73 CNR2 (0.43) CYP1A2CYP3A4TSHRHSD17B10CCNC
SCHEMBL197276 0.73 ALDH1A1 (0.37) CYP1A2CYP3A4TSHRSMN1; SMN2HSD17B10
SCHEMBL2040290 0.72 MAP4K1 (0.36) IDH1PIM1
SCHEMBL853306 0.71 TDO2 (0.49) TDO2CYP1A2CYP3A4TSHRSMN1; SMN2
SCHEMBL38095 0.71 IDH1 (0.35) IDH1
SCHEMBL1461869 0.71 CYP11B2 (0.48) TDO2CYP1A2CYP3A4TSHRSMN1; SMN2
SCHEMBL182711 0.70 PLD1 (0.53) CYP1A2CYP3A4TSHRSMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000023444-A1 5,7-DISUBSTITUTED-4-AMINOPYRIDO[2,3-D]PYRIMIDINE COMPOUNDS ABBOTT LABORATORIES (US) 2000-04-27 WO claimed
WO-2000023444-A1 5,7-DISUBSTITUTED-4-AMINOPYRIDO[2,3-D]PYRIMIDINE COMPOUNDS ABBOTT LABORATORIES (US) 2000-04-27 WO disclosed