SCHEMBL8235805

SCHEMBL8235805

COc1cc(CCC(=O)N2CCOCC2)cc(-n2c(C)cc(C(C)=O)c2-c2ccccc2)c1OC

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 3/20 0.50
HPGD P15428 2/20 0.50
HSD17B10 Q99714 2/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50
KMT2A Q03164 4/20 0.48
MEN1 O00255 2/20 0.48
FKBP1A P62942 2/20 0.45
POLB P06746 1/20 0.43
HTT P42858 1/20 0.41
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39
LMNA P02545 1/20 0.39
PTGS2 P35354 1/20 0.39
PCNA P12004 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3494085 0.82 ALDH1A1 (0.40) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL3494924 0.73 KMT2A (0.45) ALDH1A1KDM4EHPGDKMT2APOLB
SCHEMBL8236282 0.71 PDE4B (0.40) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL3496056 0.70 CA1 (0.40) KMT2AMEN1POLBLMNA
SCHEMBL4984950 0.69 CA1 (0.41) KMT2AMEN1POLBLMNA
SCHEMBL3495080 0.67 NOTUM (0.45) ALDH1A1KDM4EHPGDMAPK1
SCHEMBL3494052 0.67 NOTUM (0.55) ALDH1A1HPGDKMT2AMEN1MAPT
SCHEMBL8327592 0.66 FKBP1A (1.00) ALDH1A1HPGDKMT2AMEN1FKBP1A
SCHEMBL8328048 0.66 KMT2A (0.68) KDM4EHPGDKMT2AMEN1FKBP1A
SCHEMBL2948248 0.65 FKBP1A (0.57) ALDH1A1KDM4EHPGDHSD17B10CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed