SCHEMBL8235877

SCHEMBL8235877

O=C(O)c1c(-c2ccccc2)c(C2=CCCC=C2)nn1Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GRN P28799 2/20 0.37
SORT1 Q99523 2/20 0.37
POLB P06746 2/20 0.36
GAA P10253 1/20 0.36
LMNA P02545 1/20 0.36
GLA P06280 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HTR7 P34969 2/20 0.35
HTR1A P08908 1/20 0.35
HTR2A P28223 1/20 0.35
SLC16A3 O15427 1/20 0.35
PTGER4 P35408 1/20 0.35
KCNK3 O14649 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3494751 0.81 ALDH1A1 (0.52) ALDH1A1MEN1KMT2APOLBGAA
SCHEMBL3494459 0.69 AOC2 (0.41) ALDH1A1MEN1KMT2AGAALMNA
SCHEMBL3492508 0.67 F2RL3 (0.61) ALDH1A1MEN1KMT2APOLBGAA
SCHEMBL7778046 0.67 PTGS2 (0.52) HTR7HTR1AHTR2A
SCHEMBL7777766 0.67 HTR7 (0.48) HTR7HTR1AHTR2A
SCHEMBL7778202 0.67 PTGS2 (0.60) MEN1KMT2ASMN1; SMN2
SCHEMBL7773087 0.66 PTGS2 (0.48) KMT2ALMNA
SCHEMBL8890615 0.63 HTT (0.51) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL5441403 0.62 POLB (0.49) ALDH1A1MEN1KMT2AGRNSORT1
SCHEMBL4682097 0.61 PTGDR2 (0.51) PTGER4KCNK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed