SCHEMBL8239496

SCHEMBL8239496

Cc1[nH]c2ccccc2c1CCn1ccn(CC2CCNCC2)c1=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.46
ALDH1A1 P00352 3/20 0.46
TSHR P16473 1/20 0.46
MAOA P21397 1/20 0.42
KDM4E B2RXH2 3/20 0.42
POLB P06746 1/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTR6 P50406 1/20 0.41
KCNH2 Q12809 2/20 0.41
HDAC1 Q13547 2/20 0.41
MAPT P10636 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
CYP3A4 P08684 1/20 0.39
GRIN2C Q14957 1/20 0.38
PABPC1 P11940 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13304544 0.78 ALDH1A1 (0.42) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL10957254 0.77 ALDH1A1 (0.55) HTTALDH1A1TSHRMAOAKDM4E
SCHEMBL13304480 0.76 HDAC6 (0.52) KCNH2HDAC1
SCHEMBL13304543 0.76 GRIN2C (0.46) HTTALDH1A1TSHRKDM4ESMN1; SMN2
SCHEMBL10119912 0.72 HTT (0.52) HTTALDH1A1TSHRMAOAKDM4E
SCHEMBL10119876 0.69 MAOA (0.52) HTTALDH1A1TSHRMAOAKDM4E
SCHEMBL12154389 0.69 LMNA (0.48) HTTALDH1A1TSHRMAOAKDM4E
SCHEMBL14074159 0.67 MAPT (0.57) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL26508424 0.67 HTR2A (0.68) HTTALDH1A1TSHRKDM4EPOLB
SCHEMBL28788491 0.66 HTT (0.56) HTTALDH1A1TSHRKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899325-B1 IMIDAZOLINONE AND HYDANTOINE DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE JANSSEN PHARMACEUTICA NV (BE) 2011-11-16 EP disclosed
WO-2006136553-A1 IMIDAZOLINONE AND HYDANTOINE DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE JANSSEN PHARMACEUTICA N.V. (BE) 2006-12-28 WO disclosed