SCHEMBL8240202

SCHEMBL8240202

Cc1ccc(S(=O)(=O)C2CCCCc3c(F)ccc(F)c32)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.41
ALDH1A1 P00352 6/20 0.39
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
ACHE P22303 1/20 0.35
TP53 P04637 2/20 0.35
POLB P06746 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PTGS2 P35354 2/20 0.35
LMNA P02545 2/20 0.34
CASP6 P55212 1/20 0.34
ATM Q13315 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PTGS1 P23219 1/20 0.34
ADORA3 P0DMS8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1362911 0.88 MAPT (0.42) MAPTALDH1A1CYP3A4ACHETP53
SCHEMBL1364594 0.83 ALDH1A1 (0.37) MAPTALDH1A1CYP3A4ACHEPOLB
SCHEMBL8231615 0.79 ACHE (0.38) ALDH1A1CYP3A4TSHRACHEMEN1
SCHEMBL14441565 0.71 PTGS2 (0.38) ALDH1A1TSHRACHEMEN1KMT2A
SCHEMBL12147265 0.68 PSEN1 (0.39) ALDH1A1ACHEPOLBMEN1KMT2A
SCHEMBL14441566 0.68 PSEN1 (0.39) ALDH1A1ACHEPOLBMEN1KMT2A
SCHEMBL12147254 0.68 PSEN1 (0.39) ALDH1A1ACHEPOLBMEN1KMT2A
SCHEMBL1365544 0.68 PSEN1 (0.40) ALDH1A1CYP3A4ACHEPOLBMEN1
SCHEMBL12147236 0.68 DRD2 (0.40) MAPTALDH1A1TP53LMNA
SCHEMBL11399286 0.68 MAPT (0.44) MAPTALDH1A1CYP3A4TSHRACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007084595-A2 CARBOCYCLIC AND HETEROCYCLIC ARYLSULFONES AS GAMMA SECRETASE INHIBITORS SCHERING CORPORATION (US) 2007-07-26 WO disclosed