Methylatropine

Methylatropine

SCHEMBL824874

C[N+]1(C)C2CCC1CC(OC(=O)C(CO)c1ccccc1)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 7/20 1.00
BLM P54132 4/20 0.97
PABPC1 P11940 2/20 0.97
SMN1; SMN2 Q16637 2/20 0.89
CYP2C19 P33261 1/20 0.82
CHRM1 P11229 6/20 0.80
CHRM5 P08912 5/20 0.80
CHRM3 P20309 5/20 0.80
CHRM4 P08173 4/20 0.80
MEN1 O00255 3/20 0.80
KMT2A Q03164 3/20 0.80
TSHR P16473 2/20 0.80
CYP3A4 P08684 1/20 0.72
CYP2C9 P11712 1/20 0.72
HIF1A Q16665 1/20 0.72
HSD17B10 Q99714 1/20 0.72
KDM4E B2RXH2 1/20 0.67
LMNA P02545 1/20 0.67
POLB P06746 1/20 0.67
ADRA2C P18825 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methylatropine SCHEMBL34463463 1.00 CHRM2 (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19
Methylatropine SCHEMBL1321572 0.99 BLM (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19
Methylatropine SCHEMBL30647266 0.99 BLM (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19
Methylatropine SCHEMBL29389879 0.99 PABPC1 (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19
Methylatropine SCHEMBL30003811 0.94 SMN1; SMN2 (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19
Methylatropine SCHEMBL20798247 0.94 SMN1; SMN2 (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19
Methylatropine SCHEMBL56394 0.94 SMN1; SMN2 (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19
Atropine Oxide SCHEMBL98985 0.90 CYP2C19 (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19
Atropine Oxide SCHEMBL29369999 0.90 CYP2C19 (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19
Atropine Oxide SCHEMBL162929 0.90 CYP2C19 (1.00) CHRM2BLMPABPC1SMN1; SMN2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 163 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523944-A1 COMPOUNDS AND COMPOSITIONS FOR COGNITION-ENHANCEMENT, METHODS OF MAKING, AND METHODS OF TREATING Mithridion, Inc. (US) 2012-11-21 EP claimed
EP-2403340-A1 COMPOUNDS AND COMPOSITIONS FOR COGNITION-ENHANCEMENT, METHODS OF MAKING, AND METHODS OF TREATING Mithridion, Inc. (US) 2012-01-11 EP claimed
US-20110263613-A1 COMPOUNDS AND COMPOSITIONS FOR COGNITION-ENHANCEMENT, METHODS OF MAKING, AND METHODS OF TREATING MAPLIGHT THERAPEUTICS, INC. 2011-10-27 US claimed
WO-2011085406-A1 COMPOUNDS AND COMPOSITIONS FOR COGNITION-ENHANCEMENT, METHODS OF MAKING, AND METHODS OF TREATING MITHRIDION, INC. (US) 2011-07-14 WO claimed
WO-2010102218-A1 COMPOUNDS AND COMPOSITIONS FOR COGNITION-ENHANCEMENT, METHODS OF MAKING, AND METHODS OF TREATING MITHRIDION, INC. (US) 2010-09-10 WO claimed
EP-1438001-A4 COMPOSITIONS AND METHODS FOR INHIBITING ECCRINE PERSPIRATION IN HUMANS LUKACSKO ALISON B (US) 2006-03-15 EP claimed
EP-1438001-A2 COMPOSITIONS AND METHODS FOR INHIBITING ECCRINE PERSPIRATION IN HUMANS Lukacsko, Alison B. (US) 2004-07-21 EP claimed
US-20030064040-A1 Compositions and methods for inhibiting eccrine perspiration in humans LIGHTHOUSE INNOVATIONS, LLC 2003-04-03 US claimed
WO-2003026585-A2 COMPOSITIONS AND METHODS FOR INHIBITING ECCRINE PERSPIRATION IN HUMANS LUKACSKO ALISON B (US) 2003-04-03 WO claimed
WO-2000020414-A9 PIPERIDYLOXADIAZOLES AS DOPAMINE RECEPTOR ANTAGONISTS COMBICHEM INC (US) 2002-08-22 WO claimed
JP-H09503491-A 1997-04-08 JP claimed
EP-0314444-B1 Novel oxathiolanes and derivatives thereof, pharmaceutical compositions containing them and the use thereof as medicaments ISRAEL STATE (IL) 1996-05-29 EP claimed
EP-0711292-A1 AZA SPIRO COMPOUNDS ACTING ON THE CHOLINERGIC SYSTEM WITH MUSCARINIC AGONIST ACTIVITY KOSMIN, Gerald, Emmanuel (GB) 1996-05-15 EP claimed
EP-0303391-B1 Optical isomers of a spiroquinuclidine derivative ISRAEL STATE (IL) 1995-06-07 EP claimed
WO-1995003303-A2 AZA SPIRO COMPOUNDS ACTING ON THE CHOLINERGIC SYSTEM WITH MUSCARINIC AGONIST ACTIVITY STATE OF ISRAEL, REPRESENTED BY THE PRIME MINISTER'S OFFICE, ISRAEL INSTITUTE FOR BIOLOGICAL RESEARCH (IL) 1995-02-02 WO claimed
US-5106831-A Cholinergic agent STATE OF ISRAEL, REPRESENTED BY THE PRIME MINISTER'S OFFICE, ISRAEL INSTITUTE FOR BIOLOGICAL RESEARCH (IL) 1992-04-21 US claimed
EP-0452101-A2 Spiro bridged and unbridged heterocyclic compounds ISRAEL INSTITUTE FOR BIOLOGICAL RESEARCH (IL) 1991-10-16 EP claimed
US-5053412-A Central nervous system disorders ISRAEL INSTITUTE FOR BIOLOGICAL RESEARCH (IL) 1991-10-01 US claimed
US-4876260-A NERVOUS SYSTEM DISORDERS STATE OF ISRAEL, ISRAEL INSTITUTE OF BIOLOGICAL RESEARCH (IL) 1989-10-24 US claimed
EP-0314444-A2 Novel oxathiolanes and derivatives thereof, pharmaceutical compositions containing them and the use thereof as medicaments State of IsraelRepresented by the Prime Minister's OfficeThe Israel Institute for Biological Research (IL) 1989-05-03 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110263613-A1 COMPOUNDS AND COMPOSITIONS FOR COGNITION-ENHANCEMENT, METHODS OF MAKING, AND METHODS OF TREATING CHRM3, ACHE, CHRM4 CHRM2 6/4885BLM 1402/4885PABPC1 4851/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.