SCHEMBL8249688

SCHEMBL8249688

Nc1cc(-c2ccccc2)c[n+]([O-])c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.50
HSD17B10 Q99714 3/20 0.44
CYP3A4 P08684 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA9 Q16790 3/20 0.39
CA12 O43570 2/20 0.39
ALDH1A1 P00352 5/20 0.38
PARP1 P09874 1/20 0.37
MAPT P10636 5/20 0.35
HPGD P15428 4/20 0.35
KDM4E B2RXH2 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
LMNA P02545 2/20 0.35
ALOX15 P16050 2/20 0.35
USP2 O75604 1/20 0.35
HSP90AA1 P07900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5776467 0.75 ALDH1A1 (0.44) TDP1CA1CA2CA9CA12
SCHEMBL3741855 0.71 KMO (0.53) PARP1MEN1KMT2ATSHR
SCHEMBL4267156 0.69 MAOA (0.67) MAOAHSD17B10CYP3A4TAAR1TDP1
SCHEMBL15837471 0.69 MAOA (0.67) MAOAHSD17B10CYP3A4TAAR1TDP1
SCHEMBL3995431 0.69 MAOA (0.67) MAOAHSD17B10CYP3A4TAAR1TDP1
SCHEMBL14396437 0.69 MAOA (0.74) MAOAHSD17B10CYP3A4TAAR1TDP1
SCHEMBL1585710 0.69 L3MBTL1 (0.50) CA1CA2CA9CA12ALDH1A1
SCHEMBL16519820 0.67 HSD17B10 (0.65) MAOAHSD17B10CYP3A4TAAR1TDP1
SCHEMBL173011 0.67 MAOA (1.00) MAOAHSD17B10CYP3A4TAAR1TDP1
SCHEMBL18678323 0.67 HSD17B10 (0.65) MAOAHSD17B10CYP3A4TAAR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-B1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS BIAL PORTELA & CA SA (PT) 2015-05-27 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed