SCHEMBL8250436

SCHEMBL8250436

CCc1[nH]c2ccccc2c1CC(Cc1c(CC)[nH]c2ccccc12)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 2/20 0.47
MAPT P10636 2/20 0.47
GAA P10253 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 2/20 0.43
HPGD P15428 2/20 0.43
TSHR P16473 2/20 0.43
CYP2C19 P33261 2/20 0.43
MTNR1A P48039 2/20 0.43
MTNR1B P49286 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
MEN1 O00255 1/20 0.43
CYP2C9 P11712 1/20 0.43
KMT2A Q03164 1/20 0.43
EGFR P00533 1/20 0.42
FOLH1 Q04609 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7047345 0.86 MAPT (0.51) ALDH1A1KDM4EMAPTGAACASP1
SCHEMBL7047346 0.86 MAPT (0.51) ALDH1A1KDM4EMAPTGAACASP1
SCHEMBL3743077 0.80 KDM4E (0.67) ALDH1A1KDM4EMAPTGAACASP1
SCHEMBL27733137 0.80 KDM4E (0.44) ALDH1A1KDM4EMAPTGAACASP1
SCHEMBL27361702 0.80 CHRNB2 (0.49) ALDH1A1KDM4EMAPTGAACASP1
Hydrochloric Acid SCHEMBL28521562 0.79 KDM4E (0.65) ALDH1A1KDM4EMAPTGAACASP1
SCHEMBL6882102 0.79 HTT (0.55) ALDH1A1KDM4EMAPTGAACASP1
Water SCHEMBL11540986 0.77 HTT (0.53) ALDH1A1KDM4EMAPTGAACASP1
SCHEMBL5459223 0.76 ALDH1A1 (0.50) ALDH1A1KDM4EMAPTGAACASP1
SCHEMBL10685190 0.75 KDM4E (0.64) ALDH1A1KDM4EMAPTGAACASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991645-A1 BIS-INDOLE DERIVATIVES HAVING ANTIMETASTATIC ACTIVITY, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Roche Diagnostics GmbH (DE) 2000-04-12 EP disclosed
WO-1999000381-A1 BIS-INDOLE DERIVATIVES HAVING ANTIMETASTATIC ACTIVITY, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ROCHE DIAGNOSTICS GMBH (DE) 1999-01-07 WO disclosed