SCHEMBL8250559

SCHEMBL8250559

N#Cc1cccc(N2CCN(C(=O)c3cccnc3F)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 2/20 0.51
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPK1 P28482 2/20 0.47
HTT P42858 1/20 0.46
DRD2 P14416 2/20 0.46
DRD3 P35462 1/20 0.46
AOC3 Q16853 1/20 0.46
GPR6 P46095 3/20 0.45
USP2 O75604 2/20 0.45
TSHR P16473 1/20 0.45
MLYCD O95822 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NOTUM Q6P988 1/20 0.44
PHGDH O43175 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8247829 0.87 USP2 (0.53) SLC6A7ALDH1A1KDM4EL3MBTL1MEN1
SCHEMBL4722342 0.81 MEN1 (0.71) ALDH1A1KDM4EL3MBTL1MEN1KMT2A
SCHEMBL8246614 0.81 ALDH1A1 (0.62) ALDH1A1KMT2AHTTTSHRSMN1; SMN2
SCHEMBL1870288 0.81 SLC6A7 (0.52) SLC6A7MEN1KMT2AMAPK1HTT
SCHEMBL4718989 0.79 ALDH1A1 (0.53) ALDH1A1KDM4EL3MBTL1MEN1KMT2A
SCHEMBL8247070 0.78 SMN1; SMN2 (0.72) SLC6A7ALDH1A1KDM4EL3MBTL1MEN1
SCHEMBL4763376 0.78 SLC6A7 (0.48) SLC6A7ALDH1A1MEN1KMT2AGPR6
SCHEMBL4719103 0.78 ABL1 (0.55) ALDH1A1KDM4EL3MBTL1MAPK1HTT
SCHEMBL4722869 0.76 AKR1C3 (0.58) ALDH1A1KDM4EL3MBTL1MEN1KMT2A
SCHEMBL4766135 0.76 USP2 (0.57) SLC6A7ALDH1A1KDM4EL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007009635-A1 PHENYL SUBSTITUTED PIPERAZINE-DERIVATIVES AS INHIBITORS OF PLAMINOGENIC ACTIVATOR INHIBITORS-I (PAI-I) BAYER HEALTHCARE AG (DE) 2007-01-25 WO disclosed