SCHEMBL8263374

SCHEMBL8263374

COCCCOc1cc(CO)ccn1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 9/20 0.45
LOX P28300 6/20 0.45
RECQL P46063 1/20 0.44
ACACB O00763 2/20 0.37
CBFB Q13951 2/20 0.34
MAOA P21397 1/20 0.33
DYRK1A Q13627 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
LNPEP Q9UIQ6 1/20 0.32
CHEK1 O14757 1/20 0.32
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10183827 0.92 LOXL2 (0.46) LOXL2LOXRECQLACACBCBFB
SCHEMBL13490772 0.85 LOXL2 (0.46) LOXL2LOXACACB
SCHEMBL4934891 0.83 LOXL2 (0.67) LOXL2LOX
SCHEMBL17752 0.80 LOXL2 (0.67) LOXL2LOXRECQLACACBCBFB
SCHEMBL29841247 0.80 LOXL2 (0.67) LOXL2LOXRECQLACACBCBFB
SCHEMBL2940362 0.79 RECQL (0.50) LOXL2LOXRECQLACACBMAOA
SCHEMBL8278931 0.77 UHRF1 (0.42) LOXL2LOXACACBNPC1RAB9A
SCHEMBL1911369 0.77 ALDH1A1 (0.36) LOXL2LOXCBFBFFAR4POLB
SCHEMBL1051073 0.76 DYRK1A (0.37) LOXL2LOXACACBDYRK1AFFAR4
SCHEMBL3072454 0.75 MTNR1A (0.42) CBFBFFAR4NPC1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100029647-A1 3,4,(5)-SUBSTITUTED TETRAHYDROPHYRIDINES NOVARTIS AG (CH) 2010-02-04 US disclosed
US-20100029647-A1 3,4,(5)-SUBSTITUTED TETRAHYDROPHYRIDINES NOVARTIS AG (CH) 2010-02-04 US disclosed
WO-2006074924-A1 3,4,(5)-SUBSTITUTED TETRAHVDROPYRIDINES NOVARTIS AG (CH) 2006-07-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100029647-A1 3,4,(5)-SUBSTITUTED TETRAHYDROPHYRIDINES REN, PAH, ACE LOXL2 4638/4885LOX 2174/4885RECQL 1272/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.