SCHEMBL8287900

SCHEMBL8287900

Fc1cc(NCC2CC3CCC(C2)N3Cc2ccc3ccccc3n2)ccc1N1CCOCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
DGAT1 O75907 1/20 0.37
HTT P42858 1/20 0.36
CXCR6 O00574 1/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
S1PR1 P21453 1/20 0.36
KDR P35968 1/20 0.36
SYK P43405 1/20 0.36
KMT2A Q03164 2/20 0.36
GAA P10253 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 3/20 0.36
TSHR P16473 3/20 0.36
ALOX15 P16050 2/20 0.36
HPGD P15428 2/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8289937 0.83 GRM2 (0.49) NPC1RAB9AHTTMAPTL3MBTL1
SCHEMBL4417838 0.81 FAAH (0.42) PDE10ANPC1RAB9ADGAT1HTT
SCHEMBL8288813 0.79 P2RX3 (0.43) NPC1RAB9AHTTMAPTL3MBTL1
SCHEMBL6253989 0.77 LDHA (0.44) NPC1RAB9AHTTKMT2AGAA
SCHEMBL8287911 0.77 MAOA (0.42) NPC1RAB9AHTTMAPTL3MBTL1
Hydrochloric Acid SCHEMBL6259317 0.77 LDHA (0.44) NPC1RAB9AHTTKMT2AGAA
SCHEMBL6267930 0.75 PDE10A (0.38) PDE10ANPC1RAB9ACXCR6ALDH1A1
SCHEMBL8278308 0.74 HTT (0.48) NPC1RAB9AHTTMAPTL3MBTL1
SCHEMBL4417835 0.73 FAAH (0.49) PDE10ANPC1RAB9ADGAT1HTT
SCHEMBL8290091 0.73 HTT (0.43) NPC1RAB9ADGAT1HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005058317-A1 GLYCINE TRANSPORTER-1 INHIBIRORS GLAXO GROUP LIMITED (GB) 2005-06-30 WO disclosed