SCHEMBL8288755

SCHEMBL8288755

COc1cc(CCOS(C)(=O)=O)c(NC(=O)OC(C)(C)C)cn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.34
MTNR1A P48039 2/20 0.34
MTNR1B P49286 2/20 0.34
AAK1 Q2M2I8 1/20 0.34
RORC P51449 1/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
CA1 P00915 3/20 0.31
CA2 P00918 3/20 0.31
CA12 O43570 2/20 0.31
CA9 Q16790 2/20 0.31
MEN1 O00255 1/20 0.31
PABPC1 P11940 1/20 0.31
KMT2A Q03164 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3944673 0.84 AAK1 (0.39) ATRMTNR1AMTNR1BAAK1RORC
SCHEMBL21591739 0.83 MTNR1B (0.41) MTNR1AMTNR1BCA1CA2CA12
SCHEMBL15812122 0.79 AAK1 (0.37) ATRMTNR1AMTNR1BAAK1MEN1
SCHEMBL3948675 0.78 BRD9 (0.35) MTNR1AMTNR1BAAK1MEN1PABPC1
SCHEMBL16307600 0.76 CYP17A1 (0.40) ATRMETAP1
SCHEMBL4463941 0.76 LMNA (0.41) CA1CA12METAP1
SCHEMBL7681674 0.75 NNMT (0.47) ATRAAK1CA1CA12CA9
SCHEMBL29713519 0.75 NNMT (0.47) ATRAAK1CA1CA12CA9
SCHEMBL18940331 0.74 POLB (0.47) MMP1MMP2MMP9MMP8MMP13
SCHEMBL31309952 0.74 ATR (0.46) ATRMTNR1ARORCCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005040168-A1 AZABENZODIAZEPINES AS PHOSPHODIESTERASE-4 INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2005-05-06 WO disclosed