SCHEMBL8289012

SCHEMBL8289012

Cc1ccc(-c2ccccc2S)cc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.44
AKR1C2 P52895 3/20 0.44
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
ALOX5AP P20292 4/20 0.42
FEN1 P39748 4/20 0.42
TNKS O95271 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
AKR1B10 O60218 2/20 0.40
AKR1C4 P17516 2/20 0.40
AKR1C1 Q04828 2/20 0.40
ACHE P22303 1/20 0.40
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40
PTPRC P08575 1/20 0.40
PTPN1 P18031 1/20 0.40
NISCH Q9Y2I1 1/20 0.39
GPR3 P46089 1/20 0.39
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17184105 0.82 MAOB (0.46) AKR1C3AKR1C2ALOX5APFEN1PTPRC
SCHEMBL28677957 0.82 HTR7 (0.46) MAPTTP53ACHEBRD4CREBBP
SCHEMBL12330295 0.82 TNKS (0.57) AKR1C3AKR1C2ALOX5APFEN1TNKS
SCHEMBL19935596 0.79 TNKS (0.54) AKR1C3AKR1C2ALOX5APFEN1TNKS
SCHEMBL27363344 0.79 TNKS (0.43) AKR1C3AKR1C2MAPTTP53ALOX5AP
SCHEMBL15314774 0.78 TNKS (0.42) AKR1C3AKR1C2MAPTTP53ALOX5AP
SCHEMBL29280128 0.78 PTPRC (0.43) ALOX5APFEN1PTPRCPTPN1PTGS1
SCHEMBL28609832 0.78 ALDH1A1 (0.40) MAPTTP53AR
SCHEMBL10091244 0.76 PGR (0.44) AKR1C3AKR1C2ALOX5APFEN1TNKS
SCHEMBL22149192 0.76 BRD4 (0.44) AKR1C3AKR1C2ALOX5APFEN1TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005032490-A2 CYCLIC DIAMINES AND DERIVATIVES AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-04-14 WO disclosed