SCHEMBL8290785

SCHEMBL8290785

CC(=O)Nc1sc(C(C)=O)c(C)c1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.58
HPGD P15428 3/20 0.58
TSHR P16473 1/20 0.54
HSD17B10 Q99714 2/20 0.50
GAA P10253 2/20 0.49
KDM4E B2RXH2 2/20 0.49
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
POLB P06746 3/20 0.45
RXFP1 Q9HBX9 3/20 0.44
PRKCZ Q05513 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CISD2 Q8N5K1 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2807303 0.91 ALDH1A1 (0.60) ALDH1A1HPGDTSHRHSD17B10GAA
SCHEMBL8289563 0.83 ALDH1A1 (0.84) ALDH1A1HPGDTSHRHSD17B10GAA
SCHEMBL21612947 0.81 ALDH1A1 (0.61) ALDH1A1HPGDTSHRGAALMNA
Cyclohexane SCHEMBL7825607 0.77 ABCC1 (0.57) ALDH1A1HPGDLMNATP53NPSR1
SCHEMBL3490918 0.77 ALDH1A1 (0.59) ALDH1A1HPGDTSHRGAAKDM4E
SCHEMBL8055683 0.73 ALDH1A1 (0.60) ALDH1A1HPGDTSHRHSD17B10GAA
SCHEMBL3130253 0.72 GPR35 (0.43) ALDH1A1HPGDHSD17B10LMNATP53
SCHEMBL3066973 0.72 ALDH1A1 (0.62) ALDH1A1HPGDHSD17B10GAAKDM4E
SCHEMBL8705267 0.71 GRIN2C (0.40) ALDH1A1HPGDTSHRHSD17B10TP53
SCHEMBL11344627 0.70 ALDH1A1 (1.00) ALDH1A1HPGDTSHRHSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed