SCHEMBL8290905

SCHEMBL8290905

COC(=O)N(C)c1cccc2cc(C3CCNCC3)oc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
HTR2C P28335 3/20 0.34
CYP1A2 P05177 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CRBN Q96SW2 1/20 0.34
ADORA2A P29274 2/20 0.32
CYP1A1 P04798 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8290904 0.81 ACHE (0.46) BCHEACHEMAOAMAOBCYP1A2
SCHEMBL10906155 0.74 MAOA (0.56) BCHEACHEMAOAMAOBHTR2C
SCHEMBL8300839 0.73 ASAH1 (0.37) BCHEACHEHTR2CCYP1A2KDM4E
SCHEMBL2593078 0.70 BCHE (0.59) BCHEACHEMAOAMAOBHTR2C
SCHEMBL28792307 0.64 SLC6A2 (0.53) CYP1A2KDM4EMEN1NPC1ALDH1A1
SCHEMBL29876774 0.64 SLC6A2 (0.53) CYP1A2KDM4EMEN1NPC1ALDH1A1
SCHEMBL721717 0.64 ACHE (1.00) BCHEACHEMAOAMAOBSLC6A2
SCHEMBL2090835 0.64 SIGMAR1 (0.61) ALDH1A1HSD17B10
Citric Acid SCHEMBL7968886 0.63 BCHE (0.41) BCHEACHEMAOAMAOBHTR2C
SCHEMBL28792227 0.63 MAOA (0.44) BCHEACHEMAOAMAOBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708007-A ACETYLCHOLINESTERASE INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1998-01-13 US claimed
EP-0637586-B1 2-(Piperidin-4-yl, pyridin-4-yl and tetrahydropyridin-4-yl)-benzofuran-7-carbamate derivatives, their preparation and their use as acetylcholinesterase inhibitors HOECHST MARION ROUSSEL INC (US) 1999-06-02 EP disclosed
US-5708007-A ACETYLCHOLINESTERASE INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1998-01-13 US disclosed
EP-0637586-A1 2-(Piperidin-4-yl, pyridin-4-yl and tetrahydropyridin-4-yl)benzofuran-7-ol and carbamate derivatives, their preparation and their use as acetylcholinesterase inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1995-02-08 EP disclosed