SCHEMBL8294658

SCHEMBL8294658

CNC(=S)c1cccc(CN2CCN(C(=O)OC(C)(C)C)CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 2/20 0.49
ABCB1 P08183 1/20 0.46
KDM1A O60341 2/20 0.45
TBK1 Q9UHD2 1/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 2/20 0.44
GAA P10253 1/20 0.44
VEGFA P15692 1/20 0.44
EGLN1 Q9GZT9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8294657 0.89 GLS (0.50) GLSABCB1TBK1CYP2D6CYP2C9
SCHEMBL30525131 0.85 MEN1 (0.53) GLSTBK1CYP2D6CYP2C9CYP3A4
SCHEMBL1020384 0.85 MEN1 (0.53) GLSTBK1CYP2D6CYP2C9CYP3A4
SCHEMBL4836517 0.85 CYP2D6 (0.60) GLSABCB1CYP2D6CYP2C9MEN1
SCHEMBL8616309 0.85 GLS (0.50) GLSTBK1CYP2D6CYP2C9MEN1
SCHEMBL5570335 0.85 GLS (0.49) GLSKDM1ATBK1CYP2D6CYP2C9
SCHEMBL1022120 0.83 GLS (0.49) GLSTBK1MEN1KMT2ALMNA
SCHEMBL5571027 0.82 FAAH (0.56) GLSTBK1CYP2D6CYP2C9MEN1
SCHEMBL4837787 0.80 GLS (0.54) GLSKDM1ATBK1MEN1KMT2A
SCHEMBL8540779 0.80 ALDH1A1 (0.63) GLSKDM1ACYP2D6CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005023812-A2 PIPERAZINES AS OXYTOCIN AGONISTS FERRING B.V. (NL) 2005-03-17 WO disclosed