SCHEMBL8296809

SCHEMBL8296809

CN(C)S(=O)(=O)c1cc(N)c(N)cc1-n1ccc(=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
PKM P14618 2/20 0.34
CYP3A4 P08684 2/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MCOLN3 Q8TDD5 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
PDE2A O00408 1/20 0.31
PDE5A O76074 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300289 0.84 ALDH1A1 (0.51) ALDH1A1CA12CA1CA2CA9
SCHEMBL8437635 0.78 PKM (0.38) ALDH1A1PKMPOLB
SCHEMBL8291585 0.78 CA12 (0.37) ALDH1A1CA12CA1CA2CA9
SCHEMBL8291602 0.68 CA12 (0.36) ALDH1A1CA12CA1CA2CA9
SCHEMBL8296289 0.68 CA12 (0.36) ALDH1A1CA12CA1CA2CA9
SCHEMBL29451695 0.68 ALDH1A1 (0.52) ALDH1A1PKMCYP3A4MEN1POLB
SCHEMBL8292037 0.65 GRIA1 (0.44) ALDH1A1CA12CA1CA2CA9
SCHEMBL8291724 0.65 KDM4E (0.47) ALDH1A1CA12CA1CA2CA9
SCHEMBL16364899 0.63 ALDH1A1 (0.55) ALDH1A1PKMCYP3A4MEN1POLB
SCHEMBL1439407 0.62 GAA (0.58) ALDH1A1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676397-B1 Oxopyridinylquinoxaline derivatives SHIONOGI & CO (JP) 1999-10-20 EP disclosed
US-5677305-A NERVOUS SYSTEM DISORDERS SHIONOGI & CO., LTD. (JP) 1997-10-14 US disclosed
EP-0676397-A1 Oxopyridinylquinoxaline derivatives SHIONOGI & CO., LTD. (JP) 1995-10-11 EP disclosed