SCHEMBL8300289

SCHEMBL8300289

CN(C)S(=O)(=O)c1cc([N+](=O)[O-])c(N)cc1-n1ccc(=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
POLB P06746 2/20 0.51
PKM P14618 1/20 0.51
HTT P42858 2/20 0.41
CYP3A4 P08684 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MCOLN3 Q8TDD5 1/20 0.41
ALOX15 P16050 2/20 0.39
VCAM1 P19320 1/20 0.39
PDE2A O00408 1/20 0.39
PDE5A O76074 1/20 0.39
NFKB1 P19838 1/20 0.39
APEX1 P27695 1/20 0.39
PDE4A P27815 1/20 0.39
BLM P54132 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8296809 0.84 ALDH1A1 (0.41) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL8291560 0.75 MAPT (0.57) ALDH1A1MEN1KMT2APOLBCYP3A4
SCHEMBL8292026 0.75 MAPT (0.44) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL29451638 0.74 ALDH1A1 (0.59) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL7212568 0.74 ALDH1A1 (0.59) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL8298291 0.73 ALDH1A1 (0.64) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL8296403 0.72 ALDH1A1 (0.42) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL8291563 0.72 MAPT (0.41) ALDH1A1MEN1KMT2APOLBHTT
SCHEMBL8437635 0.70 PKM (0.38) ALDH1A1POLBPKMKDM4ELMNA
SCHEMBL8291585 0.70 CA12 (0.37) ALDH1A1POLBPKMCYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676397-B1 Oxopyridinylquinoxaline derivatives SHIONOGI & CO (JP) 1999-10-20 EP disclosed
US-5677305-A NERVOUS SYSTEM DISORDERS SHIONOGI & CO., LTD. (JP) 1997-10-14 US disclosed
EP-0676397-A1 Oxopyridinylquinoxaline derivatives SHIONOGI & CO., LTD. (JP) 1995-10-11 EP disclosed