SCHEMBL8297900

SCHEMBL8297900

CC(=O)Nc1nc2c(s1)CC(CC(=O)N1CCC(F)C1)CC2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.44
RAB9A P51151 6/20 0.42
NPC1 O15118 6/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
ALDH1A1 P00352 8/20 0.42
MAPT P10636 6/20 0.40
LMNA P02545 4/20 0.40
TDP1 Q9NUW8 2/20 0.40
TP53 P04637 3/20 0.38
HSD17B10 Q99714 1/20 0.38
PIK3CG P48736 2/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPK1 P28482 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HTT P42858 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8296502 0.82 DPP4 (0.47) DPP4
SCHEMBL8296975 0.79 TP53 (0.42) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL4864281 0.78 DPP4 (0.73) DPP4RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL21568238 0.69 RAB9A (0.52) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL1506579 0.69 PDK1 (0.58) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL1028052 0.69 PDK1 (0.58) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL1028051 0.69 PDK1 (0.58) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL7312903 0.69 NPC1 (0.54) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL1033064 0.69 RAB9A (0.54) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL12805774 0.69 RAB9A (0.54) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004112701-A2 CYCLOHEXYLGLYCINE DERIVATIVES AS DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES MERCK & CO., INC. (US) 2004-12-29 WO disclosed