SCHEMBL8299902

SCHEMBL8299902

COc1ccc(OC(F)(F)F)cc1C(=O)Nc1c[nH]nc1-c1nc2c([nH]1)CCC(CN1CCOCC1)=C2

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.38
KCNH2 Q12809 1/20 0.38
KDR P35968 2/20 0.38
LCLAT1 Q6UWP7 3/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.35
GPR6 P46095 1/20 0.35
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
RUNX1 Q01196 1/20 0.35
FOXO1 Q12778 1/20 0.35
WNT3A P56704 1/20 0.34
PDE4B Q07343 1/20 0.34
AURKA O14965 1/20 0.34
JAK2 O60674 1/20 0.34
JAK3 P52333 1/20 0.34
FGFR3 P22607 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305625 0.87 GAA (0.40) ALDH1A1PDCD1CD274
SCHEMBL8305570 0.86 CNR2 (0.39) ABL1KCNH2WNT3A
SCHEMBL12303916 0.82 KCNH2 (0.42) ABL1KCNH2KDRALDH1A1RUNX1
SCHEMBL8302364 0.81 HIF1A (0.47) ALDH1A1CD274AURKA
SCHEMBL16471209 0.78 MAPK14 (0.39) ALDH1A1KMT2A
SCHEMBL8305595 0.78 PARP1 (0.34) KCNH2ALDH1A1GPR6PDCD1CD274
SCHEMBL8300908 0.77 MAPT (0.36) PDCD1CD274AURKAJAK2JAK3
SCHEMBL8306105 0.76 PKM (0.40) KCNH2ALDH1A1
SCHEMBL13545093 0.76 AURKA (0.41) ABL1KCNH2KDRKMT2AAURKA
SCHEMBL8299878 0.75 NPC1 (0.42) ABL1KMT2AAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005002552-A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASES INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2005-01-13 WO disclosed