SCHEMBL8305595

SCHEMBL8305595

O=C(Nc1c[nH]nc1-c1nc2c([nH]1)CCC(CN1CCOCC1)=C2)c1cccc2c1OCC2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.34
MCHR1 Q99705 1/20 0.34
CCR8 P51685 1/20 0.33
KCNH2 Q12809 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
AURKA O14965 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CDK2 P24941 1/20 0.33
AURKB Q96GD4 1/20 0.33
GPR6 P46095 1/20 0.32
BCL3 P20749 3/20 0.32
POLB P06746 1/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306105 0.88 PKM (0.40) CCR8KCNH2MAPTTSHRSMN1; SMN2
SCHEMBL8305625 0.86 GAA (0.40) MAPTTSHRSMN1; SMN2BCL3POLB
SCHEMBL8300908 0.85 MAPT (0.36) PARP1MCHR1MAPTTSHRNPC1
SCHEMBL8305570 0.84 CNR2 (0.39) KCNH2BCL3
SCHEMBL8302364 0.82 HIF1A (0.47) MCHR1MAPTSMN1; SMN2AURKACDK1
SCHEMBL8302374 0.81 KDM4E (0.34) MCHR1AURKACDK1CCNB1CDK2
SCHEMBL12252752 0.81 AURKA (0.45) PARP1NPC1RAB9ASMN1; SMN2AURKA
SCHEMBL14311682 0.79 AURKA (0.43) MCHR1TSHRNPC1RAB9ASMN1; SMN2
SCHEMBL12027127 0.79 ADORA3 (0.35) MCHR1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL8299878 0.78 NPC1 (0.42) MCHR1MAPTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005002552-A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASES INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2005-01-13 WO disclosed