SCHEMBL8305625

SCHEMBL8305625

COc1ccccc1C(=O)Nc1c[nH]nc1-c1nc2c([nH]1)CCC(CN1CCOCC1)=C2

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
MAPK1 P28482 2/20 0.40
BRPF1 P55201 1/20 0.40
POLB P06746 1/20 0.40
ALDH1A1 P00352 5/20 0.40
STAT3 P40763 1/20 0.40
MAPT P10636 2/20 0.39
ALOX15 P16050 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
BCL3 P20749 2/20 0.39
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
TSHR P16473 3/20 0.38
HCN4 Q9Y3Q4 1/20 0.38
BCHE P06276 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305570 0.90 CNR2 (0.39) BCL3
SCHEMBL8299902 0.87 ABL1 (0.38) ALDH1A1PDCD1CD274
SCHEMBL8305595 0.86 PARP1 (0.34) GAAPOLBALDH1A1MAPTSMN1; SMN2
SCHEMBL8300908 0.84 MAPT (0.36) MAPTSMN1; SMN2PDCD1CD274TSHR
SCHEMBL8306105 0.84 PKM (0.40) GAAALDH1A1MAPTSMN1; SMN2BCL3
SCHEMBL8302364 0.82 HIF1A (0.47) GAAPOLBALDH1A1STAT3MAPT
SCHEMBL16471209 0.81 MAPK14 (0.39) MAPK1ALDH1A1MAPTSMN1; SMN2TSHR
SCHEMBL8299878 0.80 NPC1 (0.42) MAPK1MAPTSMN1; SMN2
SCHEMBL8302374 0.80 KDM4E (0.34)
SCHEMBL14311682 0.80 AURKA (0.43) GAAPOLBSMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005002552-A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASES INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2005-01-13 WO disclosed