SCHEMBL8305570

SCHEMBL8305570

O=C(Nc1c[nH]nc1-c1nc2c([nH]1)CCC(CN1CCOCC1)=C2)c1ccccc1OC(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.39
RXFP1 Q9HBX9 2/20 0.39
WNT3A P56704 9/20 0.38
ABL1 P00519 1/20 0.36
KCNH2 Q12809 1/20 0.36
CNR1 P21554 1/20 0.35
SLC6A9 P48067 1/20 0.35
OPRM1 P35372 1/20 0.35
BCL3 P20749 1/20 0.34
HCN1 O60741 1/20 0.34
ACKR3 P25106 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305625 0.90 GAA (0.40) BCL3
SCHEMBL8299902 0.86 ABL1 (0.38) WNT3AABL1KCNH2
SCHEMBL8302364 0.85 HIF1A (0.47)
SCHEMBL8305595 0.84 PARP1 (0.34) KCNH2BCL3
SCHEMBL8300908 0.83 MAPT (0.36)
SCHEMBL8306105 0.81 PKM (0.40) KCNH2BCL3
SCHEMBL1646552 0.80 AURKA (0.46) RXFP1WNT3AABL1KCNH2ACKR3
SCHEMBL8299878 0.79 NPC1 (0.42) ABL1
SCHEMBL8302374 0.78 KDM4E (0.34) CNR2
SCHEMBL14311682 0.78 AURKA (0.43) ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005002552-A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASES INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2005-01-13 WO disclosed