SCHEMBL8300908

SCHEMBL8300908

O=C(Nc1c[nH]nc1-c1nc2c([nH]1)CCC(CN1CCOCC1)=C2)c1cccc2nccnc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.36
HSD17B10 Q99714 1/20 0.36
IRAK4 Q9NWZ3 3/20 0.36
FGFR3 P22607 2/20 0.35
LMNA P02545 1/20 0.34
ESR1 P03372 1/20 0.34
PDCD1 Q15116 2/20 0.34
CD274 Q9NZQ7 2/20 0.34
AURKA O14965 2/20 0.33
AURKB Q96GD4 2/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CDK2 P24941 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
PARP1 P09874 2/20 0.33
MCHR1 Q99705 1/20 0.33
TAS2R8 Q9NYW2 1/20 0.33
TSHR P16473 1/20 0.33
CCKBR P32239 2/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305595 0.85 PARP1 (0.34) MAPTPDCD1CD274AURKAAURKB
SCHEMBL8305625 0.84 GAA (0.40) MAPTPDCD1CD274TSHRSMN1; SMN2
SCHEMBL8305570 0.83 CNR2 (0.39)
SCHEMBL8306105 0.82 PKM (0.40) MAPTIRAK4LMNATSHRSMN1; SMN2
SCHEMBL8305065 0.81 AURKA (0.45) MAPTHSD17B10IRAK4FGFR3AURKA
SCHEMBL8302364 0.80 HIF1A (0.47) MAPTCD274AURKAAURKBCDK1
SCHEMBL8302374 0.78 KDM4E (0.34) HSD17B10AURKAAURKBCDK1CCNB1
SCHEMBL14311682 0.78 AURKA (0.43) HSD17B10FGFR3AURKAAURKBCDK1
SCHEMBL8299878 0.77 NPC1 (0.42) MAPTAURKAAURKBCDK1CCNB1
SCHEMBL8299902 0.77 ABL1 (0.38) FGFR3PDCD1CD274AURKAJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005002552-A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASES INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2005-01-13 WO disclosed