SCHEMBL8299252

SCHEMBL8299252

CCCCCCCCOc1cc2c(c(F)n1)C(F)(F)C(c1ccc(O)cn1)CC2

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR5A1 Q13285 1/20 0.32
DEGS1 O15121 1/20 0.31
CNR2 P34972 9/20 0.31
CNR1 P21554 6/20 0.31
GPR84 Q9NQS5 1/20 0.31
STS P08842 5/20 0.30
HTR3E A5X5Y0 1/20 0.30
HTR3B O95264 1/20 0.30
HTR3A P46098 1/20 0.30
HTR3D Q70Z44 1/20 0.30
HTR3C Q8WXA8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8293940 0.90 THRA (0.35) CNR2CNR1GPR84
SCHEMBL8293978 0.88 CNR2 (0.32) CNR2CNR1GPR84
SCHEMBL8423689 0.83 MAPT (0.30)
SCHEMBL8303039 0.79 NR5A1 (0.33) NR5A1DEGS1CNR2CNR1HTR3E
SCHEMBL8301428 0.78 THRA (0.34) NR5A1DEGS1CNR2CNR1GPR84
SCHEMBL8305404 0.70 GPR84 (0.32) NR5A1CNR2CNR1GPR84HTR3E
SCHEMBL8298273 0.69 GPR84 (0.34) CNR2CNR1GPR84HTR3EHTR3B
SCHEMBL8301529 0.69 HTR1D (0.36) NR5A1CNR2CNR1GPR84
SCHEMBL8299021 0.68 NR5A1 (0.37) NR5A1DEGS1GPR84
SCHEMBL8299691 0.66 RAB9A (0.44) NR5A1DEGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828716-B1 TRIFLUORTETRAHYDRO-ISOQUINOLINE DERIVATIVES AND THE USE THEREOF IN LIQUID CRYSTALLINE MIXTURES AVENTIS RES & TECH GMBH & CO (DE) 1999-12-01 EP disclosed
US-5904877-A CHEMICAL, THERMAL AND LIGHT STABILITY HOECHST AKTIENGESELLSCHAFT (DE) 1999-05-18 US disclosed