SCHEMBL8301428

SCHEMBL8301428

CCCCCCCCOc1cc2c(c(F)n1)C(=O)C(c1ccc(O)cn1)CC2

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
GPR84 Q9NQS5 3/20 0.33
NR5A1 Q13285 1/20 0.32
HTR3E A5X5Y0 2/20 0.32
HTR3B O95264 2/20 0.32
HTR3A P46098 2/20 0.32
HTR3D Q70Z44 2/20 0.32
HTR3C Q8WXA8 2/20 0.32
DEGS1 O15121 1/20 0.31
CNR2 P34972 10/20 0.31
CNR1 P21554 7/20 0.31
TAOK3 Q9H2K8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8298273 0.88 GPR84 (0.34) THRATHRBGPR84HTR3EHTR3B
SCHEMBL8440460 0.83 MAPT (0.30)
SCHEMBL8294020 0.81 THRA (0.38) THRATHRBGPR84HTR3EHTR3B
SCHEMBL8303039 0.79 NR5A1 (0.33) NR5A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL8299252 0.78 NR5A1 (0.32) GPR84NR5A1HTR3EHTR3BHTR3A
SCHEMBL8305404 0.70 GPR84 (0.32) GPR84NR5A1HTR3EHTR3BHTR3A
SCHEMBL8293978 0.69 CNR2 (0.32) GPR84CNR2CNR1
SCHEMBL8302527 0.68 NPC1 (0.34) THRATHRB
SCHEMBL8390797 0.67 FFAR4 (0.35) THRATHRBGPR84HTR3EHTR3B
SCHEMBL8293940 0.67 THRA (0.35) THRATHRBGPR84CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824521-B1 1-FLUOR-6,7-DIHYDRO-5H-ISOQUINOLINE-8-ONE-DERIVATIVES AND THE USE THEREOF IN LIQUID CRYSTALLINE MIXTURES AVENTIS RES & TECH GMBH & CO (DE) 1999-12-01 EP disclosed
US-5874023-A ELECTROOPTICS, DISPLAYS HOECHST AKTIENGESELLSCHAFT (DE) 1999-02-23 US disclosed
EP-0824521-A1 1-FLUOR-6,7-DIHYDRO-5H-ISOQUINOLINE-8-ONE-DERIVATIVES AND THE USE THEREOF IN LIQUID CRYSTALLINE MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-25 EP disclosed
WO-1996035673-A1 1-FLUOR-6,7-DIHYDRO-5H-ISOQUINOLINE-8-ONE-DERIVATIVES AND THE USE THEREOF IN LIQUID CRYSTALLINE MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1996-11-14 WO disclosed