SCHEMBL8303058

SCHEMBL8303058

C=CCc1c(N2CCCC2=N)ccc2c1OCC(=O)N2

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.34
HTR1A P08908 3/20 0.34
NR3C2 P08235 1/20 0.33
DRD3 P35462 8/20 0.33
DRD4 P21917 7/20 0.33
HTR2A P28223 4/20 0.33
DRD1 P21728 3/20 0.33
KDM4E B2RXH2 1/20 0.31
HTR1D P28221 2/20 0.31
HTR1B P28222 2/20 0.31
SLC6A4 P31645 2/20 0.31
KCNH2 Q12809 2/20 0.31
DRD5 P21918 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL427031 0.76 MMP12 (0.39) DRD2HTR1ANR3C2DRD3DRD4
SCHEMBL8307023 0.69 DRD2 (0.38) DRD2HTR1ANR3C2DRD3DRD4
SCHEMBL8302748 0.67 DRD2 (0.39) DRD2HTR1ADRD3DRD4HTR2A
SCHEMBL426861 0.66 SMYD3 (0.43) DRD2HTR1AHTR1DHTR1BSLC6A4
SCHEMBL8304724 0.65 DRD2 (0.34) DRD2NR3C2DRD3DRD4HTR2A
SCHEMBL428017 0.65 MMP12 (0.40) DRD2HTR1ANR3C2DRD3DRD4
SCHEMBL7854062 0.65 KDM4E (0.36) NR3C2KDM4E
SCHEMBL8303552 0.64 DRD2 (0.33) DRD2HTR1A
SCHEMBL8301874 0.62 DRD2 (0.37) DRD2HTR1ANR3C2DRD3DRD4
SCHEMBL8303055 0.62 DRD2 (0.37) DRD2HTR1ANR3C2DRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0548254-B1 6- OR 7-(IMIDAZOLIDIN-2-YLIDENEAMINO)-1,4-BENZOXAZINES AS ALPHA ADRENERGIC AGENTS ALLERGAN INC (US) 1999-06-02 EP disclosed
US-5091528-A Antiglaucoma, antidiarrhea agents, diuretics, vasoconstrictors ALLERGAN, INC. (US) 1992-02-25 US disclosed