SCHEMBL8303074

SCHEMBL8303074

FC(F)(F)c1cc(-c2ccn[c]n2)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.37
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
RXRA P19793 3/20 0.35
RXRB P28702 3/20 0.35
RXRG P48443 2/20 0.35
KIF11 P52732 1/20 0.34
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
KMO O15229 1/20 0.33
F2RL3 Q96RI0 1/20 0.32
IDO1 P14902 1/20 0.32
IKBKB O14920 1/20 0.32
NOS3 P29474 1/20 0.32
NOS2 P35228 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
NISCH Q9Y2I1 1/20 0.31
TRPV3 Q8NET8 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1435833 0.71 KDM1A (0.37) KDM1AS1PR1S1PR3RXRARXRB
SCHEMBL194461 0.70 NISCH (0.33) KIF11NOS3NOS2NISCH
SCHEMBL3597375 0.69 RAB9A (0.41)
SCHEMBL19258816 0.68 NOS3 (0.52) KDM1AS1PR1S1PR3RXRARXRB
SCHEMBL30090584 0.67 NPC1 (0.52) KDM1ATDP1
SCHEMBL4577045 0.67 NPC1 (0.52) KDM1ATDP1
SCHEMBL2753599 0.67 CTSS (0.41) KDM1AS1PR1S1PR3RXRARXRB
SCHEMBL4455134 0.67 KMO (0.44) KDM1AS1PR1S1PR3KMONOS3
SCHEMBL9482063 0.66 RXRA (0.54) S1PR1S1PR3RXRARXRBRXRG
SCHEMBL990825 0.66 CYP2A6 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937051-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS & COMPANY INCORPORATED (US) 1999-08-25 EP claimed
WO-1998020003-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-05-14 WO claimed
EP-0937051-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS & COMPANY INCORPORATED (US) 1999-08-25 EP disclosed
WO-1998020003-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-05-14 WO disclosed