SCHEMBL8303462

SCHEMBL8303462

NCC(=O)Nn1cccc1C(=O)c1ccccc1F

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
ALDH1A1 P00352 6/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PTPN1 P18031 1/20 0.37
ERCC5 P28715 1/20 0.37
FEN1 P39748 1/20 0.37
GAA P10253 1/20 0.36
KAT6A Q92794 1/20 0.36
ALOX15 P16050 1/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 1/20 0.35
HPGD P15428 3/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL10365922 0.99 CES2 (0.37) CES2CES1ALDH1A1L3MBTL1PTPN1
Bromide SCHEMBL8305746 0.99 CES2 (0.37) CES2CES1ALDH1A1L3MBTL1PTPN1
Bromide SCHEMBL8305743 0.99 CES2 (0.37) CES2CES1ALDH1A1L3MBTL1PTPN1
SCHEMBL10365425 0.86 ALDH1A1 (0.39) CES2CES1ALDH1A1PTPN1ERCC5
SCHEMBL10365541 0.86 CES2 (0.38) CES2CES1ALDH1A1PTPN1ERCC5
SCHEMBL8309075 0.84 GAA (0.41) CES2CES1ALDH1A1PTPN1ERCC5
SCHEMBL8441148 0.84 GABRP (0.48) CES2CES1ALDH1A1ERCC5FEN1
SCHEMBL8308215 0.83 LMNA (0.41) GAAKAT6ARAB9A
Bromide SCHEMBL10365170 0.83 GAA (0.40) CES2CES1ALDH1A1PTPN1ERCC5
SCHEMBL10365264 0.83 CES2 (0.42) CES2CES1ALDH1A1PTPN1ERCC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582182-B1 1-Aminoacetamidopyrroles and 1-amino-2-(substituted) pyrroles and their use for the treatment of neurodegenerative dysfunctions HOECHST MARION ROUSSEL INC (US) 1999-10-20 EP claimed
US-4588727-A ANALGESICS, TRANQUILLIZERS, ANTICONVULSANTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-05-13 US claimed