SCHEMBL8303695

SCHEMBL8303695

Cc1c(N2CCNC2=N)ccc2c1OCCN2

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DRD2 P14416 2/20 0.34
HTR1A P08908 1/20 0.34
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301928 0.84 DRD2 (0.34) DRD2HTR1AAR
SCHEMBL8307985 0.83 DRD2 (0.34) DRD2HTR1A
SCHEMBL8306164 0.81 DRD2 (0.33) DRD2HTR1A
SCHEMBL8301874 0.80 DRD2 (0.37) DRD2HTR1AAR
SCHEMBL8303552 0.79 DRD2 (0.33) DRD2HTR1A
SCHEMBL8303888 0.78 ADRA2A (0.42) ALDH1A1GAAMAPTHSD17B10
SCHEMBL10027765 0.74 ALDH1A1 (0.44) ALDH1A1GAAMAPTHSD17B10DRD2
SCHEMBL8308098 0.73 ALDH1A1 (0.43) ALDH1A1GAAMAPTHSD17B10AR
SCHEMBL8307056 0.73 ALDH1A1 (0.43) ALDH1A1GAAMAPTHSD17B10AR
SCHEMBL8307073 0.69 CYP11B1 (0.32) ALDH1A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0548254-B1 6- OR 7-(IMIDAZOLIDIN-2-YLIDENEAMINO)-1,4-BENZOXAZINES AS ALPHA ADRENERGIC AGENTS ALLERGAN INC (US) 1999-06-02 EP disclosed
EP-0548254-A1 6- or 7- (2-IMINO-2-IMIDAZOLIDINE)-1,4-BENZOXAZINES AS ALPHA ADRENERGIC AGENTS ALLERGAN, INC. (US) 1993-06-30 EP disclosed
WO-1992004345-A1 6- or 7- (2-IMINO-2-IMIDAZOLIDINE)-1,4-BENZOXAZINES AS ALPHA ADRENERGIC AGENTS ALLERGAN, INC. (US) 1992-03-19 WO disclosed
US-5091528-A Antiglaucoma, antidiarrhea agents, diuretics, vasoconstrictors ALLERGAN, INC. (US) 1992-02-25 US disclosed