SCHEMBL8300039

SCHEMBL8300039

O=C(O)COCC1(O)CCC(C2CCN(Nc3ccncc3)CC2)CC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.40
ITGA2B P08514 13/20 0.40
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
GRIN2B Q13224 1/20 0.37
HSD11B1 P28845 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
AVPR1A P37288 1/20 0.32
BCHE P06276 1/20 0.32
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306140 0.74 KDM4E (0.39) ITGB3ITGA2BCYP2D6CYP2C9GRIN2B
SCHEMBL8302338 0.73 ITGB3 (0.42) ITGB3ITGA2BCYP2D6CYP2C9GRIN2B
SCHEMBL8619225 0.73 HIF1A (0.33) ITGB3ITGA2BCYP2D6CYP2C9GRIN2B
SCHEMBL8304068 0.72 CYP2D6 (0.39) ITGB3ITGA2BCYP2D6CYP2C9GRIN2B
SCHEMBL8303601 0.72 HRH3 (0.44) ITGB3ITGA2BCYP2C9
SCHEMBL8300260 0.68 ITGB3 (0.38) ITGB3ITGA2BCYP2D6CYP2C9GRIN2B
SCHEMBL30267426 0.65 EPHX1 (0.44) ITGB3ITGA2BCYP2D6CYP2C9GRIN2B
SCHEMBL8300331 0.64 KDM4E (0.43) ITGB3ITGA2BCYP2D6CYP2C9GRIN2B
SCHEMBL8300007 0.63 HSD11B1 (0.32) ITGB3ITGA2BHSD11B1
SCHEMBL8303817 0.61 KDM4E (0.40) ITGB3ITGA2BBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed