SCHEMBL8306140

SCHEMBL8306140

O=C(O)COCC1(O)CCC(N2CCN(CCNc3ccncc3)CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
GRIN2B Q13224 1/20 0.37
TRPV6 Q9H1D0 2/20 0.36
ITGB3 P05106 6/20 0.36
ITGA2B P08514 6/20 0.36
HRH3 Q9Y5N1 1/20 0.33
TACR1 P25103 1/20 0.33
SLC6A4 P31645 1/20 0.33
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300676 0.87 KDM4E (0.42) KDM4EMEN1ALDH1A1KMT2ACYP2D6
SCHEMBL8304068 0.84 CYP2D6 (0.39) CYP2D6CYP2C9GRIN2BITGB3ITGA2B
SCHEMBL8299936 0.81 KDM4E (0.41) KDM4EMEN1ALDH1A1KMT2ACYP2D6
SCHEMBL8301126 0.80 KDM4E (0.40) KDM4EMEN1ALDH1A1KMT2ACYP2D6
SCHEMBL8303583 0.80 KDM4E (0.40) KDM4EMEN1ALDH1A1KMT2ACYP2D6
SCHEMBL8301129 0.78 TRPV6 (0.47) KDM4EMEN1ALDH1A1KMT2ATRPV6
SCHEMBL8613950 0.78 KDM4E (0.39) KDM4EMEN1ALDH1A1KMT2ACYP2D6
SCHEMBL8300030 0.77 KDM4E (0.45) KDM4EMEN1ALDH1A1KMT2ACYP2D6
SCHEMBL8303601 0.77 HRH3 (0.44) CYP2C9ITGB3ITGA2BHRH3
SCHEMBL8300039 0.74 ITGB3 (0.40) CYP2D6CYP2C9GRIN2BITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed