SCHEMBL8303601

SCHEMBL8303601

O=C(O)COCC1(O)CCC(N2CCC(Oc3ccncc3)CC2)CC1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.44
ITGB3 P05106 4/20 0.41
ITGA2B P08514 4/20 0.41
EPHX2 P34913 2/20 0.40
HRH1 P35367 1/20 0.38
CCR3 P51677 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2J2 P51589 1/20 0.38
FFAR4 Q5NUL3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306140 0.77 KDM4E (0.39) HRH3ITGB3ITGA2BCYP2C9
SCHEMBL8304068 0.77 CYP2D6 (0.39) ITGB3ITGA2BHRH1CYP2C9
SCHEMBL8300007 0.76 HSD11B1 (0.32) ITGB3ITGA2B
SCHEMBL8298757 0.76 HRH3 (0.49) HRH3ITGB3ITGA2BEPHX2CYP2C9
SCHEMBL8617676 0.74 HRH3 (0.46) HRH3EPHX2HRH1CCR3
SCHEMBL8300039 0.72 ITGB3 (0.40) ITGB3ITGA2BCYP2C9
SCHEMBL639198 0.68 EPHX2 (0.60) EPHX2CYP2C9CYP2J2
SCHEMBL7399380 0.67 ITGB3 (0.49) HRH3ITGB3ITGA2B
SCHEMBL7399382 0.67 ITGB3 (0.49) HRH3ITGB3ITGA2B
SCHEMBL7399643 0.67 HRH1 (0.57) HRH3ITGB3ITGA2BHRH1CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed