SCHEMBL8304151

SCHEMBL8304151

C=CCc1c(O)cc(O)c2c(=O)cc(-c3ccc(OC)cc3)oc12.CC=CO

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.56
PARP2 Q9UGN5 3/20 0.56
PDE5A O76074 2/20 0.56
ESR1 P03372 1/20 0.56
PDE4D Q08499 1/20 0.56
ESR2 Q92731 1/20 0.56
APP P05067 3/20 0.53
AKT1 P31749 1/20 0.53
MAOB P27338 2/20 0.52
CYP19A1 P11511 1/20 0.52
ALDH1A1 P00352 3/20 0.50
MAPK1 P28482 2/20 0.50
CDK8 P49336 2/20 0.50
CDK9 P50750 2/20 0.50
MEN1 O00255 2/20 0.50
CYP3A4 P08684 2/20 0.50
KMT2A Q03164 2/20 0.50
NPC1 O15118 1/20 0.50
USP2 O75604 1/20 0.50
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19354056 0.95 PDE5A (0.61) PARP1PARP2PDE5AESR1PDE4D
SCHEMBL5276648 0.88 ALDH1A1 (0.54) PARP1PARP2APPMAOBCYP19A1
SCHEMBL8307487 0.85 FLT3 (0.61) APPAKT1MAOBCYP19A1ALDH1A1
SCHEMBL4227433 0.83 PDE5A (0.80) PARP1PARP2PDE5AESR1PDE4D
SCHEMBL8308207 0.82 AKT1 (0.61) PARP1PARP2PDE5AESR1PDE4D
SCHEMBL19353997 0.82 PARP1 (0.65) PARP1PARP2PDE5AESR1PDE4D
SCHEMBL8429382 0.81 ALDH1A1 (0.49) PARP1PARP2APPMAOBCYP19A1
SCHEMBL8308052 0.80 MAOB (0.67) MAOBCYP19A1ALDH1A1MAPK1CDK8
SCHEMBL19354052 0.79 FLT3 (0.67) AKT1MAOBCYP19A1ALDH1A1MAPK1
SCHEMBL19354126 0.77 PARP1 (0.60) PARP1PARP2PDE5AESR1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709383-B1 Diosmetin derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1999-12-15 EP disclosed
EP-0709383-A1 Diosmetin derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-05-01 EP disclosed