SCHEMBL8304916

SCHEMBL8304916

CCOC(=O)CCc1cc(CCNC(=O)OC(C)(C)C)cc(Cc2ncc[nH]2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
P2RY12 Q9H244 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
KDM4E B2RXH2 2/20 0.36
POLB P06746 2/20 0.36
NPSR1 Q6W5P4 3/20 0.35
MAPT P10636 3/20 0.35
AKT1 P31749 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GFER P55789 1/20 0.35
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PTGER4 P35408 1/20 0.34
GLA P06280 1/20 0.34
KMT2A Q03164 1/20 0.34
HTT P42858 1/20 0.33
BCHE P06276 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8309155 0.83 CYP17A1 (0.47) CA1CA2KDM4EPOLBMAPT
SCHEMBL8304739 0.81 TBXAS1 (0.46) PDE3BPDE3AP2RY12KDM4EMAPT
SCHEMBL8308082 0.80 CYP4F2 (0.41) PDE3BPDE3AP2RY12KDM4EMAPT
SCHEMBL8307372 0.80 TBXAS1 (0.53) ALDH1A1
SCHEMBL8592476 0.79 HPGD (0.42) CA1CA2POLBMAPTCYP4F2
SCHEMBL4495406 0.78 CYP4F2 (0.56) CA1CA2MAPTCYP4F2CYP4A11
SCHEMBL4713820 0.78 NPSR1 (0.47) NPSR1ALDH1A1GFERTDP1HTT
SCHEMBL11487887 0.77 TAAR1 (0.48) PDE3BPDE3AP2RY12KDM4EMAPT
SCHEMBL8308674 0.76 TBXAS1 (0.49) CA1CA2ALDH1A1GLAKMT2A
SCHEMBL11474938 0.76 CYP4F2 (0.56) PDE3BPDE3AP2RY12KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0579618-B1 PYRIDINE- AND IMIDAZOLE-DERIVED AGENTS FOR CARDIOVASCULAR DISEASES PFIZER LTD (GB) 1999-10-13 EP disclosed
US-5457118-A Pyridine derived agents for cardiovascular diseases PFIZER INC. (US) 1995-10-10 US disclosed