SCHEMBL8305010

SCHEMBL8305010

CCCCS(=O)(=O)NC1CCc2sc(C3=NNC(=O)CC3)cc2C1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.43
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
LMNA P02545 1/20 0.35
NPY1R P25929 1/20 0.35
NPY2R P49146 1/20 0.35
MAPT P10636 1/20 0.31
F2 P00734 1/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8307326 0.80 HDAC8 (0.51) HDAC8PSEN1PSEN2APH1BNCSTN
SCHEMBL8714892 0.79 HDAC8 (0.38) HDAC8PSEN1PSEN2APH1BNCSTN
SCHEMBL9414927 0.79 PNMT (0.40) HDAC8PSEN1PSEN2APH1BNCSTN
SCHEMBL8714462 0.79 HDAC8 (0.47) HDAC8PSEN1PSEN2APH1BNCSTN
SCHEMBL9383997 0.78 NR1H2 (0.35) LMNAMAPT
SCHEMBL8306283 0.77 LMNA (0.47) HDAC8PSEN1PSEN2APH1BNCSTN
SCHEMBL9414809 0.75 PDE4B (0.35)
SCHEMBL9414973 0.73 SMN1; SMN2 (0.36) LMNANPY1RNPY2RMAPT
SCHEMBL9414815 0.71 SMN1; SMN2 (0.38) HDAC8PSEN1PSEN2APH1BNCSTN
SCHEMBL9414695 0.67 PDE4B (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0579059-B1 Pyridazinone derivatives and processes for preparing the same TANABE SEIYAKU CO (JP) 1999-05-12 EP disclosed
EP-0579059-A1 Pyridazinone derivatives and processes for preparing the same TANABE SEIYAKU CO., LTD. (JP) 1994-01-19 EP disclosed